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19 Results  for Everything (Includes Articles)

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1
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Collective synthesis of natural products by means of organocascade catalysis

Jones, Spencer B ; Simmons, Bryon ; Mastracchio, Anthony ; Macmillan, David W C

Nature, 13 July 2011, Vol.475(7355), pp.183-8 [Peer Reviewed Journal]

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Direct and enantioselective {alpha}-allylation of ketones via singly occupied molecular orbital (SOMO) catalysis

Mastracchio, Anthony ; Warkentin, Alexander A ; Walji, Abbas M ; Macmillan, David W C

Proceedings of the National Academy of Sciences of the United States of America, 30 November 2010, Vol.107(48), pp.20648-51 [Peer Reviewed Journal]

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Enantioselective organocatalysis using SOMO activation

Beeson, Teresa D ; Mastracchio, Anthony ; Hong, Jun-Bae ; Ashton, Kate ; Macmillan, David W C

Science (New York, N.Y.), 27 April 2007, Vol.316(5824), pp.582-5 [Peer Reviewed Journal]

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Palladium-Catalyzed Coupling of Vinylogous Amides with Aryl Halides: Applications to the Synthesis of Heterocycles
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Palladium-Catalyzed Coupling of Vinylogous Amides with Aryl Halides: Applications to the Synthesis of Heterocycles

Edmondson, Scott D. ; Mastracchio, Anthony ; Parmee, Emma R.

Organic Letters, 04/2000, Vol.2(8), pp.1109-1112 [Peer Reviewed Journal]

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Crystal structure of human phosphodiesterase 3B: atomic basis for substrate and inhibitor specificity

Scapin, Giovanna ; Patel, Sangita B ; Chung, Christine ; Varnerin, Jeffrey P ; Edmondson, Scott D ; Mastracchio, Anthony ; Parmee, Emma R ; Singh, Suresh B ; Becker, Joseph W ; Van Der Ploeg, Lex H T ; Tota, Michael R

Biochemistry, 25 May 2004, Vol.43(20), pp.6091-100 [Peer Reviewed Journal]

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(2S,3S)-3-Amino-4-(3,3-difluoropyrrolidin-1-yl)-N,N-dimethyl-4-oxo-2-(4-1,2,4triazolo1,5-a-pyridin-6-ylphenyl)butanamide: a selective alpha-amino amide dipeptidyl peptidase IV inhibitor for the treatment of type 2 diabetes

Edmondson, Scott D ; Mastracchio, Anthony ; Mathvink, Robert J ; He, Jiafang ; Harper, Bart ; Park, You-Jung ; Beconi, Maria ; Di Salvo, Jerry ; Eiermann, George J ; He, Huaibing ; Leiting, Barbara ; Leone, Joseph F ; Levorse, Dorothy A ; Lyons, Kathryn ; Patel, Reshma A ; Patel, Sangita B ; Petrov, Aleksandr ; Scapin, Giovanna ; Shang, Jackie ; Roy

Journal of medicinal chemistry, 15 June 2006, Vol.49(12), pp.3614-27 [Peer Reviewed Journal]

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7
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Aminopiperidine-fused imidazoles as dipeptidyl peptidase-IV inhibitors

Edmondson, Scott D ; Mastracchio, Anthony ; Cox, Jason M ; Eiermann, George J ; He, Huaibing ; Lyons, Kathryn A ; Patel, Reshma A ; Patel, Sangita B ; Petrov, Aleksandr ; Scapin, Giovanna ; Wu, Joseph K ; Xu, Shiyao ; Zhu, Bing ; Thornberry, Nancy A ; Roy, Ranabir Sinha ; Weber, Ann E

Bioorganic & Medicinal Chemistry Letters, 01 August 2009, Vol.19(15), pp.4097-4101 [Peer Reviewed Journal]

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Discovery of 3-aminopiperidines as potent, selective, and orally bioavailable dipeptidyl peptidase IV inhibitors

Cox, Jason M ; Harper, Bart ; Mastracchio, Anthony ; Leiting, Barbara ; Sinha Roy, Ranabir ; Patel, Reshma A ; Wu, Joseph K ; Lyons, Kathryn A ; He, Huaibing ; Xu, Shiyao ; Zhu, Bing ; Thornberry, Nancy A ; Weber, Ann E ; Edmondson, Scott D

Bioorganic & Medicinal Chemistry Letters, 15 August 2007, Vol.17(16), pp.4579-4583 [Peer Reviewed Journal]

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Interspecies in vitro metabolism of the phosphodiesterase‐4 (PDE4) inhibitor L‐454,560

Bateman, Kevin P. ; Trimble, Laird ; Chauret, Nathalie ; Silva, Jose ; Day, Stephen ; Macdonald, Dwight ; Dube, Daniel ; Gallant, Michel ; Mastracchio, Anthony ; Perrier, Helene ; Girard, Yves ; Nicoll‐Griffith, Deborah

Journal of Mass Spectrometry, June 2006, Vol.41(6), pp.771-780 [Peer Reviewed Journal]

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Investigation of biaryl heterocycles as inhibitors of Wee1 kinase

Mastracchio, Anthony ; Lai, Chunqiu ; Torrent, Maricel ; Bromberg, Kenneth ; Buchanan, Fritz G ; Ferguson, Debra ; Bontcheva, Velitchka ; Johnson, Eric F ; Lasko, Loren ; Maag, David ; Shoemaker, Alexander R ; Penning, Thomas D

Bioorganic & Medicinal Chemistry Letters, 15 June 2019, Vol.29(12), pp.1481-1486 [Peer Reviewed Journal]

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Design, synthesis, and biological evaluation of 8-biarylquinolines: A novel class of PDE4 inhibitors

Gallant, Michel ; Chauret, Nathalie ; Claveau, David ; Day, Stephen ; Deschênes, Denis ; Dubé, Daniel ; Huang, Zheng ; Lacombe, Patrick ; Laliberté, France ; Lévesque, Jean-François ; Liu, Susana ; Macdonald, Dwight ; Mancini, Joseph ; Masson, Paul ; Mastracchio, Anthony

Bioorganic & Medicinal Chemistry Letters, 2008, Vol.18(4), pp.1407-1412 [Peer Reviewed Journal]

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Triazolopiperazine-amides as dipeptidyl peptidase IV inhibitors: Close analogs of JANUVIA™ (sitagliptin phosphate)

Kim, Dooseop ; Kowalchick, Jennifer E ; Edmondson, Scott D ; Mastracchio, Anthony ; Xu, Jinyou ; Eiermann, George J ; Leiting, Barbara ; Wu, Joseph K ; Pryor, Kellyann D ; Patel, Reshma A ; He, Huaibing ; Lyons, Kathryn A ; Thornberry, Nancy A ; Weber, Ann E

Bioorganic & Medicinal Chemistry Letters, 2007, Vol.17(12), pp.3373-3377 [Peer Reviewed Journal]

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Discovery of potent, selective, and orally bioavailable pyridone-based dipeptidyl peptidase-4 inhibitors

Xu, Jinyou ; Wei, Lan ; Mathvink, Robert ; Edmondson, Scott D ; Mastracchio, Anthony ; Eiermann, George J ; He, Huaibing ; Leone, Joseph F ; Leiting, Barbara ; Lyons, Kathryn A ; Marsilio, Frank ; Patel, Reshma A ; Petrov, Aleksandr ; Wu, Joseph K ; Thornberry, Nancy A ; Weber, Ann E

Bioorganic & Medicinal Chemistry Letters, 2006, Vol.16(5), pp.1346-1349 [Peer Reviewed Journal]

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14
Process Development and Large-Scale Synthesis of a PDE4 Inhibitor
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Process Development and Large-Scale Synthesis of a PDE4 Inhibitor

Conlon, David A. ; Drahus-Paone, Antoinette ; Ho, Guo-Jie ; Pipik, Brenda ; Helmy, Roy ; Mcnamara, James M. ; Shi, Yao-Jun ; Williams, J. Michael ; Macdonald, Dwight ; Deschênes, Denis ; Gallant, Michel ; Mastracchio, Anthony ; Roy, Bruno ; Scheigetz, John

Organic Process Research & Development, 01/2006, Vol.10(1), pp.36-45 [Peer Reviewed Journal]

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15
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Discovery of potent and selective orally bioavailable β-substituted phenylalanine derived dipeptidyl peptidase IV inhibitors

Edmondson, Scott D ; Mastracchio, Anthony ; Duffy, Joseph L ; Eiermann, George J ; He, Huaibing ; Ita, Ida ; Leiting, Barbara ; Leone, Joseph F ; Lyons, Kathryn A ; Makarewicz, Amanda M ; Patel, Reshma A ; Petrov, Aleksandr ; Wu, Joseph K ; Thornberry, Nancy A ; Weber, Ann E

Bioorganic & Medicinal Chemistry Letters, 2005, Vol.15(12), pp.3048-3052 [Peer Reviewed Journal]

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16
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4-Amino cyclohexylglycine analogues as potent dipeptidyl peptidase IV inhibitors

Parmee, Emma R ; He, Jiafang ; Mastracchio, Anthony ; Edmondson, Scott D ; Colwell, Larry ; Eiermann, George ; Feeney, William P ; Habulihaz, Bahanu ; He, Huaibing ; Kilburn, Ruth ; Leiting, Barbara ; Lyons, Kathryn ; Marsilio, Frank ; Patel, Reshma A ; Petrov, Aleksandr ; Di Salvo, Jerry ; Wu, Joseph K ; Thornberry, Nancy A ; Weber, Ann E

Bioorganic & Medicinal Chemistry Letters, 2004, Vol.14(1), pp.43-46 [Peer Reviewed Journal]

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17
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Potent and selective proline derived dipeptidyl peptidase IV inhibitors

Edmondson, Scott D ; Mastracchio, Anthony ; Beconi, Maria ; Colwell, Lawrence F ; Habulihaz, Bahanu ; He, Huaibing ; Kumar, Sanjeev ; Leiting, Barbara ; Lyons, Kathryn A ; Mao, Ann ; Marsilio, Frank ; Patel, Reshma A ; Wu, Joseph K ; Zhu, Lan ; Thornberry, Nancy A ; Weber, Ann E ; Parmee, Emma R

Bioorganic & Medicinal Chemistry Letters, 18 October 2004, Vol.14(20), pp.5151-5155 [Peer Reviewed Journal]

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Discovery of a substituted 8-arylquinoline series of PDE4 inhibitors: Structure–activity relationship, optimization, and identification of a highly potent, well tolerated, PDE4 inhibitor

Macdonald, Dwight ; Mastracchio, Anthony ; Perrier, Hélène ; Dubé, Daniel ; Gallant, Michel ; Lacombe, Patrick ; Deschênes, Denis ; Roy, Bruno ; Scheigetz, John ; Bateman, Kevin ; Li, Chun ; Trimble, Laird A ; Day, Stephen ; Chauret, Nathalie ; Nicoll-Griffith, Deborah A ; Silva, Jose M

Bioorganic & Medicinal Chemistry Letters, 2005, Vol.15(23), pp.5241-5246 [Peer Reviewed Journal]

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Benzyl vinylogous amide substituted aryldihydropyridazinones and aryldimethylpyrazolones as potent and selective PDE3B inhibitors

Edmondson, Scott D ; Mastracchio, Anthony ; He, Jiafang ; Chung, Christine C ; Forrest, Michael J ; Hofsess, Scott ; Macintyre, Euan ; Metzger, Joseph ; O'Connor, Naphtali ; Patel, Kajal ; Tong, Xinchun ; Tota, Michael R ; Van Der Ploeg, Lex H.T ; Varnerin, Jeff P ; Fisher, Michael H ; Wyvratt, Matthew J ; Weber, Ann E ; Parmee, Emma R

Bioorganic & Medicinal Chemistry Letters, 2003, Vol.13(22), pp.3983-3987 [Peer Reviewed Journal]

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