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Synthesis of new 4,5-dihydrofuranoindoles and their evaluation as HCV NS5B polymerase inhibitors

Velázquez, Francisco ; Venkatraman, Srikanth ; Lesburg, Charles A ; Duca, José ; Rosenblum, Stuart B ; Kozlowski, Joseph A ; Njoroge, F George

Organic letters, 20 January 2012, Vol.14(2), pp.556-9 [Peer Reviewed Journal]

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2
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Discovery of Chromane Containing Hepatitis C Virus (HCV) NS5A Inhibitors with Improved Potency against Resistance-Associated Variants

Yu, Wensheng ; Tong, Ling ; Hu, Bin ; Zhong, Bin ; Hao, Jinglai ; Ji, Tao ; Zan, Shuai ; Coburn, Craig A ; Selyutin, Oleg ; Chen, Lei ; Rokosz, Laura ; Agrawal, Sony ; Liu, Rong ; Curry, Stephanie ; Mcmonagle, Patricia ; Ingravallo, Paul ; Asante-Appiah, Ernest ; Chen, Shiying ; Kozlowski, Joseph A

Journal of medicinal chemistry, 23 November 2016, Vol.59(22), pp.10228-10243 [Peer Reviewed Journal]

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3
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Synthesis and SAR studies of benzimidazolone derivatives as histamine H3-receptor antagonists

Zeng, Qingbei ; Rosenblum, Stuart B ; Yang, Zhaoxia ; Jiang, Yueheng ; Mccormick, Kevin D ; Aslanian, Robert G ; Duguma, Luli ; Kozlowski, Joseph A ; Shih, Neng-Yang ; Hey, John A ; West, Robert E ; Korfmacher, Walter A ; Berlin, Michael ; Boyce, Christopher W

Bioorganic & Medicinal Chemistry Letters, 01 November 2013, Vol.23(21), pp.6001-6003 [Peer Reviewed Journal]

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4
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Development of a prodrug of hydantoin based TACE inhibitor

Tong, Ling ; Kim, Seong Heon ; Chen, Lei ; Kosinski, Aneta ; Shankar, Bandarpalle B ; Girijavallabhan, Vinay ; Yang, De-Yi ; Yu, Wensheng ; Zhou, Guowei ; Shih, Neng-Yang ; Chen, Shiying ; Hu, Mengwei ; Lundell, Daniel ; Niu, Xiaoda ; Umland, Shelby ; Kozlowski, Joseph A

Bioorganic & Medicinal Chemistry Letters, 15 August 2017, Vol.27(16), pp.3704-3708 [Peer Reviewed Journal]

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5
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Selective benzylic lithiation of N-Boc-2-phenylpiperidine and pyrrolidine: expedient synthesis of a 2,2-disubstituted piperidine NK 1 antagonist

Xiao, Dong ; Lavey, Brian J ; Palani, Anandan ; Wang, Cheng ; Aslanian, Robert G ; Kozlowski, Joseph A ; Shih, Neng-Yang ; Mcphail, Andrew T ; Randolph, Gerard P ; Lachowicz, Jean E ; Duffy, Ruth A

Tetrahedron Letters, 2005, Vol.46(44), pp.7653-7656 [Peer Reviewed Journal]

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6
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Synthesis of mono- and difluoronaphthoic acids

Tagat, Jayaram R ; Mccombie, Stuart W ; Nazareno, Dennis V ; Boyle, Craig D ; Kozlowski, Joseph A ; Chackalamannil, Samuel ; Josien, Hubert ; Wang, Yuguang ; Zhou, Guowei

The Journal of organic chemistry, 22 February 2002, Vol.67(4), pp.1171-7 [Peer Reviewed Journal]

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7
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Further insight into lower order cuprate chemistry; On the use of CuBr·Me2S vs CuI enroute to R2CuLi

H. Lipshutz, Bruce ; Whitney, Scott ; Kozlowski, Joseph A ; Breneman, Curt M

Tetrahedron Letters, 1986, Vol.27(36), pp.4273-4276 [Peer Reviewed Journal]

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8
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Effects of Lewis acids on higher order, mixed cuprate couplings

Lipshutz, Bruce H ; Parker, David A ; Kozlowski, Joseph A ; Nguyen, Sam L

Tetrahedron Letters, 1984, Vol.25(52), pp.5959-5962 [Peer Reviewed Journal]

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9
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Ligand mixing in lower order organocuprates: synthetic, mechanistic, and structural implications

Lipshutz, Bruce H ; Kozlowski, Joseph A ; Breneman, Curt M

Tetrahedron Letters, 1985, Vol.26(48), pp.5911-5914 [Peer Reviewed Journal]

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10
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Alternative core development around the tetracyclic indole class of HCV NS5A inhibitors

Tong, Ling ; Yu, Wensheng ; Coburn, Craig A ; Meinke, Peter T ; Nair, Anilkumar G ; Dwyer, Michael P ; Chen, Lei ; Selyutin, Oleg ; Rosenblum, Stuart B ; Jiang, Yueheng ; Fells, James ; Hu, Bin ; Zhong, Bin ; Soll, Richard M ; Liu, Rong ; Agrawal, Sony ; Xia, Ellen ; Zhai, Ying ; Kong, Rong ; Ingravallo

Bioorganic & medicinal chemistry letters, 15 October 2016, Vol.26(20), pp.5132-5137 [Peer Reviewed Journal]

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11
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MK-8325: A silyl proline-containing NS5A inhibitor with pan-genotype activity for treatment of HCV

Nair, Anilkumar G ; Zeng, Qingbei ; Selyutin, Oleg ; Rosenblum, Stuart B ; Jiang, Yueheng ; Yang, De-Yi ; Keertikar, Kerry ; Zhou, Guowei ; Dwyer, Michael ; Kim, Seong Heon ; Shankar, Bandarpalle ; Yu, Wensheng ; Tong, Ling ; Chen, Lei ; Mazzola, Robert ; Caldwell, John ; Tang, Haiqun ; Agrawal, Sony ; Liu, Rong ; Kong

Bioorganic & medicinal chemistry letters, 01 June 2018, Vol.28(10), pp.1954-1957 [Peer Reviewed Journal]

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12
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Discovery of SCH 900188: A Potent Hepatitis C Virus NS5B Polymerase Inhibitor Prodrug As a Development Candidate

Chen, Kevin X ; Venkatraman, Srikanth ; Anilkumar, Gopinadhan N ; Zeng, Qingbei ; Lesburg, Charles A ; Vibulbhan, Bancha ; Velazquez, Francisco ; Chan, Tin-Yau ; Bennet, Frank ; Jiang, Yueheng ; Pinto, Patrick ; Huang, Yuhua ; Selyutin, Oleg ; Agrawal, Sony ; Huang, Hsueh-Cheng ; Li, Cheng ; Cheng, Kuo-Chi ; Shih, Neng-Yang ; Kozlowski, Joseph A ; Rosenblum

ACS medicinal chemistry letters, 13 March 2014, Vol.5(3), pp.244-8 [Peer Reviewed Journal]

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13
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IV. Discovery of CXCR3 antagonists substituted with heterocycles as amide surrogates: improved PK, hERG and metabolic profiles

Nair, Anilkumar G ; Wong, Michael K C ; Shu, Youheng ; Jiang, Yueheng ; Jenh, Chung-Her ; Kim, Seong Heon ; Yang, De-Yi ; Zeng, Qingbei ; Shao, Yuefei ; Zawacki, Lisa Guise ; Duo, Jingqi ; Mcguinness, Brian F ; Carroll, Carolyn Diianni ; Hobbs, Doug W ; Shih, Neng-Yang ; Rosenblum, Stuart B ; Kozlowski, Joseph A

Bioorganic & medicinal chemistry letters, 15 February 2014, Vol.24(4), pp.1085-8 [Peer Reviewed Journal]

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14
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2-(2-Aminothiazol-4-yl)pyrrolidine-based tartrate diamides as potent, selective and orally bioavailable TACE inhibitors

Dai, Chaoyang ; Li, Dansu ; Popovici-Muller, Janeta ; Zhao, Lianyun ; Girijavallabhan, Vinay M ; Rosner, Kristin E ; Lavey, Brian J ; Rizvi, Razia ; Shankar, Bandarpalle B ; Wong, Michael K.C ; Guo, Zhuyan ; Orth, Peter ; Strickland, Corey O ; Sun, Jing ; Niu, Xiaoda ; Chen, Shiying ; Kozlowski, Joseph A ; Lundell, Daniel J ; Piwinski, John J ; Shih, Neng-Yang

Bioorganic & Medicinal Chemistry Letters, 2011, Vol.21(10), pp.3172-3176 [Peer Reviewed Journal]

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15
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Fused bi-heteroaryl substituted hydantoin compounds as TACE inhibitors

Tong, Ling ; Kim, Seong Heon ; Rosner, Kristin ; Yu, Wensheng ; Shankar, Bandarpalle B ; Chen, Lei ; Li, Dansu ; Dai, Chaoyang ; Girijavallabhan, Vinay ; Popovici-Muller, Janeta ; Yang, Liping ; Zhou, Guowei ; Kosinski, Aneta ; Siddiqui, M Arshad ; Shih, Neng-Yang ; Guo, Zhuyan ; Orth, Peter ; Chen, Shiying ; Lundell, Daniel ; Niu

Bioorganic & medicinal chemistry letters, 15 July 2017, Vol.27(14), pp.3037-3042 [Peer Reviewed Journal]

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16
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III. Identification of novel CXCR3 chemokine receptor antagonists with a pyrazinyl–piperazinyl–piperidine scaffold

Kim, Seong Heon ; Anilkumar, Gopinadhan N ; Zawacki, Lisa Guise ; Zeng, Qingbei ; Yang, De-Yi ; Shao, Yuefei ; Dong, Guizhen ; Xu, Xiaolian ; Yu, Wensheng ; Jiang, Yueheng ; Jenh, Chung-Her ; Hall, James W ; Carroll, Carolyn Diianni ; Hobbs, Doug W ; Baldwin, John J ; Mcguinness, Brian F ; Rosenblum, Stuart B ; Kozlowski, Joseph A ; Shankar, Bandarpalle B ; Shih, Neng-Yang

Bioorganic & Medicinal Chemistry Letters, 2011, Vol.21(23), pp.6982-6986 [Peer Reviewed Journal]

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17
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II. SAR studies of pyridyl–piperazinyl-piperidine derivatives as CXCR3 chemokine antagonists

Shao, Yuefei ; Anilkumar, Gopinadhan N ; Carroll, Carolyn Diianni ; Dong, Guizhen ; Hall, James W ; Hobbs, Doug W ; Jiang, Yueheng ; Jenh, Chung-Her ; Kim, Seong Heon ; Kozlowski, Joseph A ; Mcguinness, Brian F ; Rosenblum, Stuart B ; Schulman, Inna ; Shih, Neng-Yang ; Shu, Youheng ; Wong, Michael K.C ; Yu, Wensheng ; Zawacki, Lisa Guise ; Zeng, Qingbei

Bioorganic & Medicinal Chemistry Letters, 2011, Vol.21(5), pp.1527-1531 [Peer Reviewed Journal]

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18
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The chemistry of higher order organocuprates

Lipshutz, Bruce H ; Wilhelm, Robert S ; Kozlowski, Joseph A

Tetrahedron, 1984, Vol.40(24), pp.5005-5038 [Peer Reviewed Journal]

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19
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Expansion of SAR studies on triaryl bis sulfone cannabinoid CB 2 receptor ligands

Tong, Ling ; Shankar, B.B ; Chen, Lei ; Rizvi, Razia ; Kelly, Joseph ; Gilbert, Eric ; Huang, Chunli ; Yang, De-Yi ; Kozlowski, Joseph A ; Shih, N.-Y ; Gonsiorek, W ; Hipkin, R. William ; Malikzay, Asra ; Lunn, Charles A ; Lundell, Daniel J

Bioorganic & Medicinal Chemistry Letters, 2010, Vol.20(22), pp.6785-6789 [Peer Reviewed Journal]

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20
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I. Novel HCV NS5B polymerase inhibitors: discovery of indole 2-carboxylic acids with C3-heterocycles

Anilkumar, Gopinadhan N ; Lesburg, Charles A ; Selyutin, Oleg ; Rosenblum, Stuart B ; Zeng, Qingbei ; Jiang, Yueheng ; Chan, Tin-Yau ; Pu, Haiyan ; Vaccaro, Henry ; Wang, Li ; Bennett, Frank ; Chen, Kevin X ; Duca, Jose ; Gavalas, Stephen ; Huang, Yuhua ; Pinto, Patrick ; Sannigrahi, Mousumi ; Velazquez, Francisco ; Venkatraman, Srikanth ; Vibulbhan

Bioorganic & medicinal chemistry letters, 15 September 2011, Vol.21(18), pp.5336-41 [Peer Reviewed Journal]

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21
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Aryl or heteroaryl substituted aminal derivatives of HCV NS5A inhibitor MK-8742

Yu, Wensheng ; Coburn, Craig A ; Nair, Anilkumar G ; Wong, Michael ; Rosenblum, Stuart B ; Zhou, Guowei ; Dwyer, Michael P ; Tong, Ling ; Hu, Bin ; Zhong, Bin ; Hao, Jinglai ; Ji, Tao ; Zan, Shuai ; Kim, Seong Heon ; Zeng, Qingbei ; Selyutin, Oleg ; Chen, Lei ; Masse, Frederic ; Agrawal, Sony ; Liu

Bioorganic & medicinal chemistry letters, 01 August 2016, Vol.26(15), pp.3414-20 [Peer Reviewed Journal]

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22
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Structure-activity relationship (SAR) development and discovery of potent indole-based inhibitors of the hepatitis C virus (HCV) NS5B polymerase

Chen, Kevin X ; Vibulbhan, Bancha ; Yang, Weiying ; Sannigrahi, Mousumi ; Velazquez, Francisco ; Chan, Tin-Yau ; Venkatraman, Srikanth ; Anilkumar, Gopinadhan N ; Zeng, Qingbei ; Bennet, Frank ; Jiang, Yueheng ; Lesburg, Charles A ; Duca, Jose ; Pinto, Patrick ; Gavalas, Stephen ; Huang, Yuhua ; Wu, Wanli ; Selyutin, Oleg ; Agrawal, Sony ; Feld

Journal of medicinal chemistry, 26 January 2012, Vol.55(2), pp.754-65 [Peer Reviewed Journal]

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23
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Discovery of MK-6169, a Potent Pan-Genotype Hepatitis C Virus NS5A Inhibitor with Optimized Activity against Common Resistance-Associated Substitutions

Yu, Wensheng ; Tong, Ling ; Selyutin, Oleg ; Chen, Lei ; Hu, Bin ; Zhong, Bin ; Hao, Jinglai ; Ji, Tao ; Zan, Shuai ; Yin, Jingjun ; Ruck, Rebecca T ; Curry, Stephanie ; Mcmonagle, Patricia ; Agrawal, Sony ; Rokosz, Laura ; Carr, Donna ; Ingravallo, Paul ; Bystol, Karin ; Lahser, Frederick ; Liu

Journal of medicinal chemistry, 10 May 2018, Vol.61(9), pp.3984-4003 [Peer Reviewed Journal]

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24
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Substituted tetracyclic indole core derivatives of HCV NS5A inhibitor MK-8742

Yu, Wensheng ; Zhou, Guowei ; Coburn, Craig A ; Zeng, Qingbei ; Tong, Ling ; Dwyer, Michael P ; Hu, Bin ; Zhong, Bin ; Hao, Jinglai ; Ji, Tao ; Zan, Shuai ; Chen, Lei ; Mazzola, Robert ; Kim, Jae-Hun ; Sha, Deyou ; Selyutin, Oleg ; Rosenblum, Stuart B ; Lavey, Brian ; Nair, Anilkumar G ; Heon Kim

Bioorganic & medicinal chemistry letters, 01 October 2016, Vol.26(19), pp.4851-4856 [Peer Reviewed Journal]

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25
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II. Novel HCV NS5B polymerase inhibitors: discovery of indole C2 acyl sulfonamides

Anilkumar, Gopinadhan N ; Selyutin, Oleg ; Rosenblum, Stuart B ; Zeng, Qingbei ; Jiang, Yueheng ; Chan, Tin-Yau ; Pu, Haiyan ; Wang, Li ; Bennett, Frank ; Chen, Kevin X ; Lesburg, Charles A ; Duca, Jose ; Gavalas, Stephen ; Huang, Yuhua ; Pinto, Patrick ; Sannigrahi, Mousumi ; Velazquez, Francisco ; Venkatraman, Srikanth ; Vibulbhan, Bancha ; Agrawal

Bioorganic & medicinal chemistry letters, 01 January 2012, Vol.22(1), pp.713-7 [Peer Reviewed Journal]

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26
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Alkyl substituted aminal derivatives of HCV NS5A inhibitor MK-8742

Yu, Wensheng ; Coburn, Craig A ; Nair, Anilkumar G ; Wong, Michael ; Tong, Ling ; Dwyer, Michael P ; Hu, Bin ; Zhong, Bin ; Hao, Jinglai ; Yang, De-Yi ; Selyutin, Oleg ; Jiang, Yueheng ; Rosenblum, Stuart B ; Kim, Seong Heon ; Lavey, Brian J ; Zhou, Guowei ; Rizvi, Razia ; Shankar, Bandarpalle B ; Zeng, Qingbei ; Chen, Lei ; Agrawal, Sony ; Carr, Donna ; Rokosz, Laura ; Liu, Rong ; Curry, Stephanie ; Mcmonagle, Patricia ; Ingravallo, Paul ; Lahser, Fred ; Asante-Appiah, Ernest ; Nomeir, Amin ; Kozlowski, Joseph A

Bioorganic & medicinal chemistry letters, 01 August 2016, Vol.26(15), pp.3800-5 [Peer Reviewed Journal]

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27
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Discovery of silyl proline containing HCV NS5A inhibitors with pan-genotype activity: SAR development

Nair, Anilkumar G ; Zeng, Qingbei ; Selyutin, Oleg ; Rosenblum, Stuart B ; Jiang, Yueheng ; Yang, De-Yi ; Keertikar, Kerry ; Zhou, Guowei ; Dwyer, Michael P ; Kim, Seong Heon ; Shankar, Bandarpalle ; Yu, Wensheng ; Tong, Ling ; Chen, Lei ; Mazzola, Robert ; Caldwell, John ; Tang, Haiqun ; Allard, Melissa L ; Buckle, Ronald N ; Gauuan

Bioorganic & medicinal chemistry letters, 01 March 2016, Vol.26(5), pp.1475-9 [Peer Reviewed Journal]

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28
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Matched and mixed cap derivatives in the tetracyclic indole class of HCV NS5A inhibitors

Dwyer, Michael P ; Keertikar, Kerry M ; Chen, Lei ; Tong, Ling ; Selyutin, Oleg ; Nair, Anilkumar G ; Yu, Wensheng ; Zhou, Guowei ; Lavey, Brian J ; Yang, De-Yi ; Wong, Michael ; Kim, Seong Heon ; Coburn, Craig A ; Rosenblum, Stuart B ; Zeng, Qingbei ; Jiang, Yueheng ; Shankar, Bandarpalle B ; Rizvi, Razia ; Nomeir, Amin A ; Liu

Bioorganic & medicinal chemistry letters, 15 August 2016, Vol.26(16), pp.4106-11 [Peer Reviewed Journal]

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29
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Discovery of 3-morpholino-imidazole1,5-apyrazine BTK inhibitors for rheumatoid arthritis

Boga, Sobhana Babu ; Alhassan, Abdul-Basit ; Liu, Jian ; Guiadeen, Deodial ; Krikorian, Arto ; Gao, Xiaolei ; Wang, James ; Yu, Younong ; Anand, Rajan ; Liu, Shilan ; Yang, Chundao ; Wu, Hao ; Cai, Jiaqiang ; Zhu, Hugh ; Desai, Jagdish ; Maloney, Kevin ; Gao, Ying-Duo ; Fischmann, Thierry O ; Presland, Jeremy ; Mansueto

Bioorganic & medicinal chemistry letters, 15 August 2017, Vol.27(16), pp.3939-3943 [Peer Reviewed Journal]

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30
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Structure-activity relationships of proline modifications around the tetracyclic-indole class of NS5A inhibitors

Tong, Ling ; Yu, Wensheng ; Coburn, Craig A ; Chen, Lei ; Selyutin, Oleg ; Zeng, Qingbei ; Dwyer, Michael P ; Nair, Anilkumar G ; Shankar, Bandarpalle B ; Kim, Seong Heon ; Yang, De-Yi ; Rosenblum, Stuart B ; Ruck, Rebecca T ; Davies, Ian W ; Hu, Bin ; Zhong, Bin ; Hao, Jinglai ; Ji, Tao ; Zan, Shuai ; Liu

Bioorganic & medicinal chemistry letters, 01 November 2016, Vol.26(21), pp.5354-5360 [Peer Reviewed Journal]

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31
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Discovery of fused tricyclic core containing HCV NS5A inhibitors with pan-genotype activity

Yu, Wensheng ; Coburn, Craig A ; Yang, De-Yi ; Meinke, Peter T ; Wong, Michael ; Rosenblum, Stuart B ; Chen, Kevin X ; Njoroge, George F ; Chen, Lei ; Dwyer, Michael P ; Jiang, Yueheng ; Nair, Anilkumar G ; Selyutin, Oleg ; Tong, Ling ; Zeng, Qingbei ; Zhong, Bin ; Ji, Tao ; Hu, Bin ; Agrawal, Sony ; Xia

Bioorganic & medicinal chemistry letters, 01 July 2016, Vol.26(13), pp.3158-3162 [Peer Reviewed Journal]

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32
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Discovery of potent macrocyclic HCV NS5A inhibitors

Yu, Wensheng ; Vibulbhan, Bancha ; Rosenblum, Stuart B ; Martin, Gregory S ; Vellekoop, A Samuel ; Holst, Christian L ; Coburn, Craig A ; Wong, Michael ; Selyutin, Oleg ; Ji, Tao ; Zhong, Bin ; Hu, Bin ; Chen, Lei ; Dwyer, Michael P ; Jiang, Yueheng ; Nair, Anilkumar G ; Tong, Ling ; Zeng, Qingbei ; Agrawal, Sony ; Carr

Bioorganic & medicinal chemistry letters, 01 August 2016, Vol.26(15), pp.3793-9 [Peer Reviewed Journal]

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33
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A novel class of highly potent irreversible hepatitis C virus NS5B polymerase inhibitors

Chen, Kevin X ; Lesburg, Charles A ; Vibulbhan, Bancha ; Yang, Weiying ; Chan, Tin-Yau ; Venkatraman, Srikanth ; Velazquez, Francisco ; Zeng, Qingbei ; Bennett, Frank ; Anilkumar, Gopinadhan N ; Duca, Jose ; Jiang, Yueheng ; Pinto, Patrick ; Wang, Li ; Huang, Yuhua ; Selyutin, Oleg ; Gavalas, Stephen ; Pu, Haiyan ; Agrawal, Sony ; Feld

Journal of medicinal chemistry, 08 March 2012, Vol.55(5), pp.2089-101 [Peer Reviewed Journal]

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34
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Characterization of peripheral human cannabinoid receptor (hCB2) expression and pharmacology using a novel radioligand, 35SSch225336

Gonsiorek, Waldemar ; Hesk, David ; Chen, Shu-Cheng ; Kinsley, David ; Fine, Jay S ; Jackson, James V ; Bober, Loretta A ; Deno, Gregory ; Bian, Hong ; Fossetta, James ; Lunn, Charles A ; Kozlowski, Joseph A ; Lavey, Brian ; Piwinski, John ; Narula, Satwant K ; Lundell, Daniel J ; Hipkin, R William

The Journal of biological chemistry, 22 September 2006, Vol.281(38), pp.28143-51 [Peer Reviewed Journal]

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35
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Non-aromatic A-ring replacement in the triaryl bis-sulfone CB2 receptor inhibitors

Gilbert, Eric J ; Zhou, Guowei ; Wong, Michael K.C ; Tong, Ling ; Shankar, Bandarpalle B ; Huang, Chunli ; Kelly, Joseph ; Lavey, Brian J ; Mccombie, Stuart W ; Chen, Lei ; Rizvi, Razia ; Dong, Youhao ; Shu, Youheng ; Kozlowski, Joseph A ; Shih, Neng-Yang ; Hipkin, R. William ; Gonsiorek, Waldemar ; Malikzay, Asra ; Lunn, Charles A ; Favreau, Len

Bioorganic & Medicinal Chemistry Letters, 2010, Vol.20(2), pp.608-611 [Peer Reviewed Journal]

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36
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Discovery of Ruzasvir (MK-8408): A Potent, Pan-Genotype HCV NS5A Inhibitor with Optimized Activity against Common Resistance-Associated Polymorphisms

Tong, Ling ; Yu, Wensheng ; Chen, Lei ; Selyutin, Oleg ; Dwyer, Michael P ; Nair, Anilkumar G ; Mazzola, Robert ; Kim, Jae-Hun ; Sha, Deyou ; Yin, Jingjun ; Ruck, Rebecca T ; Davies, Ian W ; Hu, Bin ; Zhong, Bin ; Hao, Jinglai ; Ji, Tao ; Zan, Shuai ; Liu, Rong ; Agrawal, Sony ; Xia

Journal of medicinal chemistry, 12 January 2017, Vol.60(1), pp.290-306 [Peer Reviewed Journal]

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