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Stereoselective addition of 2-phenyloxazol-4-yl trifluoromethanesulfonate to N-sulfinyl imines: application to the synthesis of the HCV protease inhibitor boceprevir

Morris, William J ; Muppalla, Kiran K ; Cowden, Cameron ; Ball, Richard G

The Journal of organic chemistry, 18 January 2013, Vol.78(2), pp.706-10 [Peer Reviewed Journal]

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Synthesis of antifungal glucan synthase inhibitors from enfumafungin

Zhong, Yong-Li ; Gauthier, Donald R ; Shi, Yao-Jun ; Mclaughlin, Mark ; Chung, John Y L ; Dagneau, Philippe ; Marcune, Benjamin ; Krska, Shane W ; Ball, Richard G ; Reamer, Robert A ; Yasuda, Nobuyoshi

The Journal of organic chemistry, 06 April 2012, Vol.77(7), pp.3297-310 [Peer Reviewed Journal]

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Preparation of 2,5,7-trithiabicyclo2.2.1heptane from 1,2-bis-triisopropylsilanylsulfanyl alkenes

Gareau, Yves ; Juteau, Hélène ; Tsou, Nancy N ; Ball, Richard G

Organic letters, 05 January 2006, Vol.8(1), pp.59-61 [Peer Reviewed Journal]

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8-Azabicyclo[3.2.1]oct-3-en-2-ones via asymmetric 1,3-dipolar cycloaddition of a homochiral 3-oxidopyridinium betaine

Curtis, Neil R ; Ball, Richard G ; Kulagowski, Janusz J

Tetrahedron Letters, 2006, Vol.47(15), pp.2635-2638 [Peer Reviewed Journal]

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2-(3aR,4R,5S,7aS)-5-{(1S)-1-3,5-bis(trifluoromethyl)phenyl-2-hydroxyethoxy}-4-(2-methylphenyl)octahydro-2H-isoindol-2-yl-1,3-oxazol-4(5H)-one: a potent human NK1 receptor antagonist with multiple clearance pathways

Kassick, Andrew J ; Jiang, Jinlong ; Bunda, Jaime ; Wilson, David ; Bao, Jianming ; Lu, Huagang ; Lin, Peter ; Ball, Richard G ; Doss, George A ; Tong, Xinchun ; Tsao, Kwei-Lan C ; Wang, Hong ; Chicchi, Gary ; Karanam, Bindhu ; Tschirret-Guth, Richard ; Samuel, Koppara ; Hora, Donald F ; Kumar, Sanjeev ; Madeira, Maria ; Eng, Waisi ; Hargreaves, Richard ; Purcell, Mona ; Gantert, Liza ; Cook, Jacquelyn ; Devita, Robert J ; Mills, Sander G

Journal of medicinal chemistry, 25 July 2013, Vol.56(14), pp.5940-8 [Peer Reviewed Journal]

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Two Novel Pharmaceutical Cocrystals of a Development Compound – Screening, Scale-up, and Characterization
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Two Novel Pharmaceutical Cocrystals of a Development Compound – Screening, Scale-up, and Characterization

Leung, Dennis H. ; Lohani, Sachin ; Ball, Richard G. ; Canfield, Nicole ; Wang, Yaling ; Rhodes, Timothy ; Bak, Annette

Crystal Growth & Design, 03/07/2012, Vol.12(3), pp.1254-1262 [Peer Reviewed Journal]

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Dipolar Cycloaddition Route to Diverse Analogues of Cocaine: The 6- and 7-Substituted 3-Phenyltropanes

Kozikowski, Alan P ; Araldi, Gian Luca ; Ball, Richard G

The Journal of organic chemistry, 07 February 1997, Vol.62(3), pp.503-509 [Peer Reviewed Journal]

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8
Synthesis of the Tetracyclic Carbon Core of Menogaril Utilizing the Benzannulation Reaction of a Fischer Carbene Complex and an Alkyne
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Synthesis of the Tetracyclic Carbon Core of Menogaril Utilizing the Benzannulation Reaction of a Fischer Carbene Complex and an Alkyne

Su, Jing ; Wulff, William D. ; Ball, Richard G.

The Journal of Organic Chemistry, 11/1998, Vol.63(23), pp.8440-8447 [Peer Reviewed Journal]

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Chemistry of platensimycin

Singh, Sheo B ; Herath, Kithsiri B ; Wang, Jun ; Tsou, Nancy ; Ball, Richard G

Tetrahedron Letters, 2007, Vol.48(31), pp.5429-5433 [Peer Reviewed Journal]

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Isolation and structure elucidation of parnafungins, antifungal natural products that inhibit mRNA polyadenylation

Parish, Craig A ; Smith, Scott K ; Calati, Kathleen ; Zink, Deborah ; Wilson, Kenneth ; Roemer, Terry ; Jiang, Bo ; Xu, Deming ; Bills, Gerald ; Platas, Gonzalo ; Peláez, Fernando ; Díez, Maria Teresa ; Tsou, Nancy ; Mckeown, Arlene E ; Ball, Richard G ; Powles, Mary Ann ; Yeung, Lai ; Liberator, Paul ; Harris, Guy

Journal of the American Chemical Society, 04 June 2008, Vol.130(22), pp.7060-6 [Peer Reviewed Journal]

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Discovery of N-(4R)-6-(4-chlorophenyl)-7-(2,4-dichlorophenyl)-2,2-dimethyl-3,4-dihydro-2H-pyrano2,3-bpyridin-4-yl-5-methyl-1H-pyrazole-3-carboxamide (MK-5596) as a novel cannabinoid-1 receptor (CB1R) inverse agonist for the treatment of obesity

Yan, Lin ; Huo, Pei ; Debenham, John S ; Madsen-Duggan, Christina B ; Lao, Julie ; Chen, Richard Z ; Xiao, Jing Chen ; Shen, Chun-Pyn ; Stribling, D Sloan ; Shearman, Lauren P ; Strack, Alison M ; Tsou, Nancy ; Ball, Richard G ; Wang, Junying ; Tong, Xinchun ; Bateman, Thomas J ; Reddy, Vijay B G ; Fong, Tung M ; Hale, Jeffrey J

Journal of medicinal chemistry, 27 May 2010, Vol.53(10), pp.4028-37 [Peer Reviewed Journal]

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12
Asymmetric Synthesis of α,α-Difluoro-β-amino Acid Derivatives from Enantiomerically Pure N-tert- Butylsulfinimines
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Asymmetric Synthesis of α,α-Difluoro-β-amino Acid Derivatives from Enantiomerically Pure N-tert- Butylsulfinimines

Staas, Donnette D. ; Savage, Kelly L. ; Homnick, Carl F. ; Tsou, Nancy N. ; Ball, Richard G.

The Journal of Organic Chemistry, 11/2002, Vol.67(23), pp.8276-8279 [Peer Reviewed Journal]

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Asymmetric synthesis of alpha,alpha-difluoro-beta-amino acid derivatives from enantiomerically pure N-tert-butylsulfinimines

Staas, Donnette D ; Savage, Kelly L ; Homnick, Carl F ; Tsou, Nancy N ; Ball, Richard G

The Journal of organic chemistry, 15 November 2002, Vol.67(23), pp.8276-9 [Peer Reviewed Journal]

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14
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Diastereoselective triple radical cyclization of a bromomethyldimethylsilyl allyl ether

Kende, Andrew S ; Journet, Michel ; Ball, Richard G ; Tsou, Nancy N

Tetrahedron Letters, 1996, Vol.37(35), pp.6295-6298 [Peer Reviewed Journal]

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15
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Diastereoselective Friedel-Crafts alkylation of indoles with chiral alpha-phenyl benzylic cations. Asymmetric synthesis of anti-1,1,2-triarylalkanes

Chung, John Y L ; Mancheno, Danny ; Dormer, Peter G ; Variankaval, Narayan ; Ball, Richard G ; Tsou, Nancy N

Organic letters, 17 July 2008, Vol.10(14), pp.3037-40 [Peer Reviewed Journal]

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16
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Isolation, structure, and absolute stereochemistry of platensimycin, a broad spectrum antibiotic discovered using an antisense differential sensitivity strategy

Singh, Sheo B ; Jayasuriya, Hiranthi ; Ondeyka, John G ; Herath, Kithsiri B ; Zhang, Chaowei ; Zink, Deborah L ; Tsou, Nancy N ; Ball, Richard G ; Basilio, Angela ; Genilloud, Olga ; Diez, Maria Teresa ; Vicente, Francisca ; Pelaez, Fernando ; Young, Katherine ; Wang, Jun

Journal of the American Chemical Society, 13 September 2006, Vol.128(36), pp.11916-20 [Peer Reviewed Journal]

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17
Isolation, Structure, and Absolute Stereochemistry of Platensimycin, A Broad Spectrum Antibiotic Discovered Using an Antisense Differential Sensitivity Strategy [ J. Am. Chem. Soc. 2006 , 128 , 11916−11920].
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Isolation, Structure, and Absolute Stereochemistry of Platensimycin, A Broad Spectrum Antibiotic Discovered Using an Antisense Differential Sensitivity Strategy [ J. Am. Chem. Soc. 2006 , 128 , 11916−11920].

Singh, Sheo B. ; Jayasuriya, Hiranthi ; Ondeyka, John G. ; Herath, Kithsiri B. ; Zhang, Chaowei ; Zink, Deborah L. ; Tsou, Nancy N. ; Ball, Richard G. ; Basilio, Angela ; Genilloud, Olga ; Diez, Maria Teresa ; Vicente, Francisca ; Pelaez, Fernando ; Young, Katherine ; Wang, Jun

Journal of the American Chemical Society, 12/2006, Vol.128(48), pp.15547-15547 [Peer Reviewed Journal]

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18
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A Spectroscopic and Crystallographic Study of Polymorphism in an Aza‐Steroid

Wenslow, Robert M ; Baum, Mary W ; Ball, Richard G ; Mccauley, James A ; Varsolona, Richard J

Journal of Pharmaceutical Sciences, November 2002, Vol.91(11), pp.2465-2465 [Peer Reviewed Journal]

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19
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The synthesis and conformational analysis of amino acid–tetrahydroanthranilic acid hybrids

Imbriglio, Jason E ; Dirocco, Daniel ; Raghavan, Subharekha ; Ball, Richard G ; Tsou, Nancy ; Mosley, Ralph T ; Tata, James R ; Colletti, Steven L

Tetrahedron Letters, 2008, Vol.49(33), pp.4897-4900 [Peer Reviewed Journal]

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20
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3-Hydroxy-4-oxo-4 H-pyrido[1,2- a]pyrimidine-2-carboxylates—fast access to a heterocyclic scaffold for HIV-1 integrase inhibitors

Kinzel, Olaf D ; Ball, Richard G ; Donghi, Monica ; Maguire, Courtney K ; Muraglia, Ester ; Pesci, Silvia ; Rowley, Michael ; Summa, Vincenzo

Tetrahedron Letters, 2008, Vol.49(46), pp.6556-6558 [Peer Reviewed Journal]

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21
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Synthesis of C 2-symmetric trans-2,6-diarylpiperidinones via aryl cuprate addition: an unexpected stereochemical outcome

Hamblett, Christopher L ; Sloman, David L ; Kliman, Laura T ; Adams, Bruce ; Ball, Richard G ; Stanton, Matthew G

Tetrahedron Letters, 2007, Vol.48(12), pp.2079-2082 [Peer Reviewed Journal]

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22
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An unusual fragmentation process discovered during the course of cleavage of a camphanic acid amide

Kozikowski, Alan P ; Chen, Chinpiao ; Ball, Richard G

Tetrahedron Letters, 1990, Vol.31(41), pp.5869-5872 [Peer Reviewed Journal]

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23
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A concise and enantioselective synthesis of novel HIV-1 protease transition state mimics

Dorsey, Bruce D ; Plzak, Kevin J ; Ball, Richard G

Tetrahedron Letters, 1993, Vol.34(12), pp.1851-1854 [Peer Reviewed Journal]

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24
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A novel synthetic approach toward the zaragozic acids core structure

Koyama, Hiroo ; Ball, Richard G ; Berger, Gregory D

Tetrahedron Letters, 1994, Vol.35(49), pp.9185-9188 [Peer Reviewed Journal]

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25
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The discovery of potent antagonists of NPBWR1 (GPR7)

Anthony Romero, F ; Hastings, Nicholas B ; Moningka, Remond ; Guo, Zhiqiang ; Wang, Ming ; Di Salvo, Jerry ; Lei, Ying ; Trusca, Dorina ; Deng, Qiaolin ; Tong, Vincent ; Terebetski, Jenna L ; Ball, Richard G ; Ujjainwalla, Feroze

Bioorganic & Medicinal Chemistry Letters, 15 January 2012, Vol.22(2), pp.1014-1018 [Peer Reviewed Journal]

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26
Careful Navigation of the Crystallographic Landscape of MK-8970: A Racemic Acetal Carbonate Prodrug of Raltegravir
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Careful Navigation of the Crystallographic Landscape of MK-8970: A Racemic Acetal Carbonate Prodrug of Raltegravir

Tsou, Nancy ; Shultz, C. Scott ; Andreani, Teresa ; Ball, Richard G. ; Brunskill, Andrew ; Balsells, Jaume ; Cohen, Ryan D. ; Dasilva, Jimmy ; Li, Jing ; Reamer, Robert A. ; de Lera Ruiz, Manuel ; Variankaval, Narayan ; Varsolona, Richard J. ; Yasuda, Nobuyoshi ; York, Gregory

Organic Process Research & Development, 12/18/2015, Vol.19(12), pp.1882-1890 [Peer Reviewed Journal]

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27
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A cascade approach to cyclic aminonitrones: reaction discovery, mechanism, and scope

Sharma, Rojita ; Bulger, Paul G ; Mcnevin, Michael ; Dormer, Peter G ; Ball, Richard G ; Streckfuss, Eric ; Cuff, James F ; Yin, Jingjun ; Chen, Cheng-Yi

Organic letters, 06 August 2009, Vol.11(15), pp.3194-7 [Peer Reviewed Journal]

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28
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Pseudo-allylic A 1,3 strain as a conformational control element: Stereoselective syntheses of ψ[CH 2O] pseudodipeptides

Anthony, Neville J ; Gomez, Robert P ; Holtz, Wilbur J ; Murphy, Joan S ; Ball, Richard G ; Lee, Ta- Jyh

Tetrahedron Letters, 1995, Vol.36(22), pp.3821-3824 [Peer Reviewed Journal]

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29
Neighboring Group Participation of the Indole Nucleus:  An Unusual DAST-Mediated Rearrangement Reaction
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Neighboring Group Participation of the Indole Nucleus:  An Unusual DAST-Mediated Rearrangement Reaction

Hallett, David J. ; Gerhard, Ute ; Goodacre, Simon C. ; Hitzel, Laure ; Sparey, Timothy J. ; Thomas, Steven ; Rowley, Michael ; Ball, Richard G.

The Journal of Organic Chemistry, 08/2000, Vol.65(16), pp.4984-4993 [Peer Reviewed Journal]

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30
Asymmetric Synthesis of a Glucagon Receptor Antagonist via Friedel–Crafts Alkylation of Indole with Chiral α-Phenyl Benzyl Cation
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Asymmetric Synthesis of a Glucagon Receptor Antagonist via Friedel–Crafts Alkylation of Indole with Chiral α-Phenyl Benzyl Cation

Chung, John Y. L. ; Steinhuebel, Dietrich ; Krska, Shane W. ; Hartner, Fred W. ; Cai, Chaoxian ; Rosen, Jonathan ; Mancheno, Danny E. ; Pei, Tao ; Dimichele, Lisa ; Ball, Richard G. ; Chen, Cheng-Yi ; Tan, Lushi ; Alorati, Antony D. ; Brewer, Sarah E. ; Scott, Jeremy P.

Organic Process Research & Development, 11/16/2012, Vol.16(11), pp.1832-1845 [Peer Reviewed Journal]

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31
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Novel transannular rearrangements of azalide iminoethers

Wilkening, Robert R ; Ratcliffe, Ronald W ; Doss, George A ; Mosley, Ralph T ; Ball, Richard G

Tetrahedron, 1997, Vol.53(50), pp.16923-16944 [Peer Reviewed Journal]

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32
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Design and synthesis of conformationally constrained N,N-disubstituted 1,4-diazepanes as potent orexin receptor antagonists

Coleman, Paul J ; Schreier, John D ; Mcgaughey, Georgia B ; Bogusky, Michael J ; Cox, Christopher D ; Hartman, George D ; Ball, Richard G ; Harrell, C. Meacham ; Reiss, Duane R ; Prueksaritanont, Thomayant ; Winrow, Christopher J ; Renger, John J

Bioorganic & Medicinal Chemistry Letters, 2010, Vol.20(7), pp.2311-2315 [Peer Reviewed Journal]

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33
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Conformational analysis and receptor docking of N-(1S,2S)-3-(4-chlorophenyl)-2-(3-cyanophenyl)-1-methylpropyl-2-methyl-2-{5-(trifluoromethyl)pyridin-2-yloxy}propanamide (taranabant, MK-0364), a novel, acyclic cannabinoid-1 receptor inverse agonist

Lin, Linus S ; Ha, Sookhee ; Ball, Richard G ; Tsou, Nancy N ; Castonguay, Laurie A ; Doss, George A ; Fong, Tung M ; Shen, Chun-Pyn ; Xiao, Jing Chen ; Goulet, Mark T ; Hagmann, William K

Journal of medicinal chemistry, 10 April 2008, Vol.51(7), pp.2108-14 [Peer Reviewed Journal]

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34
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A Cavaet on the Swern Oxidation

Smith, Amos B ; Leenay, Tamara L ; Liu, Hsing-Jang ; Lloyd A.K.Nelson ; Ball, Richard G

Tetrahedron Letters, 1988, Vol.29(1), pp.49-52 [Peer Reviewed Journal]

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35
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Stereoselective synthesis of the hydroxyethylene isostere of the HIV protease (Tyr-Pro) cleavage site

Thompson, Wayne J ; Ball, Richard G ; Darke, Paul L ; Zugay, Joan A ; Thies, J.E

Tetrahedron Letters, 1992, Vol.33(21), pp.2957-2960 [Peer Reviewed Journal]

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36
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Potent nor-triterpenoid blockers of the voltage-gated potassium channel Kv1.3 from Spachea correae

Goetz, Michael A ; Hensens, Otto D ; Zink, Deborah L ; Borris, Robert P ; Morales, Francisco ; Tamayo-Castillo, Giselle ; Slaughter, Robert S ; Felix, John ; Ball, Richard G

Tetrahedron Letters, 1998, Vol.39(19), pp.2895-2898 [Peer Reviewed Journal]

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