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1,2,3-Trisubstituted cyclohexyl substance P antagonists: significance of the ring nitrogen in piperidine-based NK-1 receptor antagonists

Mills, Sander G ; Maccoss, Malcolm ; Underwood, Dennis ; Shah, Shrenik K ; Finke, Paul E ; Miller, Daniel J ; Budhu, Richard J ; Cascieri, Margaret A ; Sadowski, Sharon ; Strader, Catherine D

Bioorganic & Medicinal Chemistry Letters, 1995, Vol.5(13), pp.1345-1350 [Peer Reviewed Journal]

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1,2,4-Triacylpiperidine substance p antagonists: Separation of affinities for the NK-1 receptor and the L-type calcium channel

Mills, Sander G ; Maccoss, Malcolm ; Cascieri, Margaret A ; Sadowski, Sharon ; Patel, Smita ; Chapman, Kerry L ; Hutson, Peter H

Bioorganic & Medicinal Chemistry Letters, 1995, Vol.5(6), pp.599-604 [Peer Reviewed Journal]

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1,3,4 Trisubstituted pyrrolidine CCR5 receptor antagonists bearing 4-aminoheterocycle substituted piperidine side chains

Willoughby, Christopher A ; Rosauer, Keith G ; Hale, Jeffery J ; Budhu, Richard J ; Mills, Sander G ; Chapman, Kevin T ; Maccoss, Malcolm ; Malkowitz, Lorraine ; Springer, Martin S ; Gould, Sandra L ; Demartino, Julie A ; Siciliano, Salvatore J ; Cascieri, Margaret A ; Carella, Anthony ; Carver, Gwen ; Holmes, Karen ; Schleif, William A ; Danzeisen, Renee ; Hazuda, Daria ; Kessler, Joseph ; Lineberger, Janet ; Miller, Michael ; Emini, Emilio A

Bioorganic & medicinal chemistry letters, 10 February 2003, Vol.13(3), pp.427-31 [Peer Reviewed Journal]

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1,3,4-Trisubstituted pyrrolidine CCR5 receptor antagonists: modifications of the arylpropylpiperidine side chains

Lynch, Christopher L ; Willoughby, Christopher A ; Hale, Jeffrey J ; Holson, Edward J ; Budhu, Richard J ; Gentry, Amy L ; Rosauer, Keith G ; Caldwell, Charles G ; Chen, Ping ; Mills, Sander G ; Maccoss, Malcolm ; Berk, Scott ; Chen, Liya ; Chapman, Kevin T ; Malkowitz, Lorraine ; Springer, Martin S ; Gould, Sandra L ; Demartino, Julie A ; Siciliano, Salvatore J ; Cascieri, Margaret A ; Carella, Anthony ; Carver, Gwen ; Holmes, Karen ; Schleif, William A ; Danzeisen, Renee ; Hazuda, Daria ; Kessler, Joseph ; Lineberger, Janet ; Miller, Michael ; Emini, Emilio A

Bioorganic & Medicinal Chemistry Letters, 2003, Vol.13(1), pp.119-123 [Peer Reviewed Journal]

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1,3,4-Trisubstituted pyrrolidine CCR5 receptor antagonists. Part 1: discovery of the pyrrolidine scaffold and determination of its stereochemical requirements

Hale, Jeffrey J ; Budhu, Richard J ; Mills, Sander G ; Maccoss, Malcolm ; Malkowitz, Lorraine ; Siciliano, Salvatore ; Gould, Sandra L ; Demartino, Julie A ; Springer, Martin S

Bioorganic & Medicinal Chemistry Letters, 2001, Vol.11(11), pp.1437-1440 [Peer Reviewed Journal]

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1,3,4-Trisubstituted pyrrolidine CCR5 receptor antagonists. Part 2: lead optimization affording selective, orally bioavailable compounds with potent Anti-HIV activity

Hale, Jeffrey J ; Budhu, Richard J ; Holson, Edward B ; Finke, Paul E ; Oates, Bryan ; Mills, Sander G ; Maccoss, Malcolm ; Gould, Sandra L ; Demartino, Julie A ; Springer, Martin S ; Siciliano, Salvatore ; Malkowitz, Lorraine ; Schleif, William A ; Hazuda, Daria ; Miller, Michael ; Kessler, Joseph ; Danzeisen, Renee ; Holmes, Karen ; Lineberger, Janet ; Carella, Anthony ; Carver, Gwen ; Emini, Emilio

Bioorganic & Medicinal Chemistry Letters, 2001, Vol.11(20), pp.2741-2745 [Peer Reviewed Journal]

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1,3,4-Trisubstituted pyrrolidine CCR5 receptor antagonists. Part 3: polar functionality and its effect on anti-HIV-1 activity

Hale, Jeffrey J ; Budhu, Richard J ; Mills, Sander G ; Maccoss, Malcolm ; Gould, Sandra L ; Demartino, Julie A ; Springer, Martin S ; Siciliano, Salvatore J ; Malkowitz, Lorraine ; Schleif, William A ; Hazuda, Daria ; Miller, Michael ; Kessler, Joseph ; Danzeisen, Renee ; Holmes, Karen ; Lineberger, Janet ; Carella, Anthony ; Carver, Gwen ; Emini, Emilio A

Bioorganic & Medicinal Chemistry Letters, 21 October 2002, Vol.12(20), pp.2997-3000 [Peer Reviewed Journal]

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1,3,4-Trisubstituted pyrrolidine CCR5 receptor antagonists. Part 4: Synthesis of N-1 acidic functionality affording analogues with enhanced antiviral activity against HIV

Lynch, Christopher L ; Hale, Jeffrey J ; Budhu, Richard J ; Gentry, Amy L ; Mills, Sander G ; Chapman, Kevin T ; Maccoss, Malcolm ; Malkowitz, Lorraine ; Springer, Martin S ; Gould, Sandra L ; Demartino, Julie A ; Siciliano, Salvatore J ; Cascieri, Margaret A ; Carella, Anthony ; Carver, Gwen ; Holmes, Karen ; Schleif, William A ; Danzeisen, Renee ; Hazuda, Daria ; Kessler, Joseph ; Lineberger, Janet ; Miller, Michael ; Emini, Emilio A

Bioorganic & Medicinal Chemistry Letters, 21 October 2002, Vol.12(20), pp.3001-3004 [Peer Reviewed Journal]

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1,4-Diacylpiperazine-2-(S)-[(N-aminoalkyl)carboxamides] as novel, potent substance P receptor antagonists

Mills, Sander G ; Wu, Mu Tsu ; Maccoss, Malcolm ; Budhu, Richard J ; Dorn, Conrad P ; Cascieri, Margaret A ; Sadowski, Sharon ; Strader, Catherine D ; Greenlee, William J

Bioorganic & Medicinal Chemistry Letters, 1993, Vol.3(12), pp.2707-2712 [Peer Reviewed Journal]

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10
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17O NMR spectroscopy of nucleoside derivatives; bonding characteristics of pyrimidine carbonyls

Schwartz, Herbert M ; Maccoss, Malcolm ; Danyluk, Steven S

Tetrahedron Letters, 1980, Vol.21(40), pp.3837-3840 [Peer Reviewed Journal]

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11
2( S )-((3,5-Bis(trifluoromethyl)benzyl)oxy)-3( S )-phenyl-4-((3-oxo-1,2,4-triazol- 5-yl)methyl)morpholine ( 1 ):  A Potent, Orally Active, Morpholine-Based Human Neurokinin-1 Receptor Antagonist
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2( S )-((3,5-Bis(trifluoromethyl)benzyl)oxy)-3( S )-phenyl-4-((3-oxo-1,2,4-triazol- 5-yl)methyl)morpholine ( 1 ):  A Potent, Orally Active, Morpholine-Based Human Neurokinin-1 Receptor Antagonist

Hale, Jeffrey J. ; Mills, Sander G. ; Maccoss, Malcolm ; Shah, Shrenik K. ; Qi, Hongbo ; Mathre, David J. ; Cascieri, Margaret A. ; Sadowski, Sharon ; Strader, Catherine D. ; Macintyre, D. Euan ; Metzger, Joseph M.

Journal of Medicinal Chemistry, 01/1996, Vol.39(9), pp.1760-1762 [Peer Reviewed Journal]

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12
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4-Amino-2-alkyl-butyramides as small molecule CCR2 antagonists with favorable pharmacokinetic properties

Butora, Gabor ; Morriello, Gregori J ; Kothandaraman, Shankaran ; Guiadeen, Deodialsingh ; Pasternak, Alexander ; Parsons, William H ; Maccoss, Malcolm ; Vicario, Pasquale P ; Cascieri, Margaret A ; Yang, Lihu

Bioorganic & Medicinal Chemistry Letters, 15 September 2006, Vol.16(18), pp.4715-4722 [Peer Reviewed Journal]

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13
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5-Benzothiazole substituted pyrimidine derivatives as HCV replication (replicase) inhibitors

Arasappan, Ashok ; Bennett, Frank ; Girijavallabhan, Vinay ; Huang, Yuhua ; Huelgas, Regina ; Alvarez, Carmen ; Chen, Lei ; Gavalas, Stephen ; Kim, Seong-Heon ; Kosinski, Aneta ; Pinto, Patrick ; Rizvi, Razia ; Rossman, Randall ; Shankar, Bandarpalle ; Tong, Ling ; Velazquez, Francisco ; Venkatraman, Srikanth ; Verma, Vishal A ; Kozlowski, Joseph ; Shih, Neng-Yang ; Piwinski, John J ; Maccoss, Malcolm ; Kwong, Cecil D ; Clark, Jeremy L ; Fowler, Anita T ; Geng, Feng ; Kezar, Hollis S ; Roychowdhury, Abhijit ; Reynolds, Robert C ; Maddry, Joseph A ; Ananthan, Subramaniam ; Secrist, John A ; Li, Cheng ; Chase, Robert ; Curry, Stephanie ; Huang, Hsueh-Cheng ; Tong, Xiao ; Njoroge, F George

Bioorganic & medicinal chemistry letters, 01 May 2012, Vol.22(9), pp.3229-34 [Peer Reviewed Journal]

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14
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A 7-deaza-adenosine analog is a potent and selective inhibitor of hepatitis C virus replication with excellent pharmacokinetic properties

Olsen, David B ; Eldrup, Anne B ; Bartholomew, Linda ; Bhat, Balkrishen ; Bosserman, Michele R ; Ceccacci, Alessandra ; Colwell, Lawrence F ; Fay, John F ; Flores, Osvaldo A ; Getty, Krista L ; Grobler, Jay A ; Lafemina, Robert L ; Markel, Eric J ; Migliaccio, Giovanni ; Prhavc, Marija ; Stahlhut, Mark W ; Tomassini, Joanne E ; Maccoss, Malcolm ; Hazuda, Daria J ; Carroll, Steven S

Antimicrobial agents and chemotherapy, October 2004, Vol.48(10), pp.3944-53 [Peer Reviewed Journal]

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15
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A facile synthesis of the novel Neurokinin A antagonist SR 48968

Hale, Jeffrey J ; Finke, Paul E ; Maccoss, Malcolm

Bioorganic & Medicinal Chemistry Letters, 1993, Vol.3(2), pp.319-322 [Peer Reviewed Journal]

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16
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A notable conversion of a thiolacetate to its corresponding sulfonyl chloride

Huang, Yuhua ; Bennett, Frank ; Verma, Vishal ; George Njoroge, F ; Maccoss, Malcolm

Tetrahedron Letters, 27 June 2012, Vol.53(26), pp.3203-3205 [Peer Reviewed Journal]

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17
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Activated ketones as potent reversible inhibitors of interleukin-Iβ converting enzyme

Mjalli, Adnan M.M ; Chapman, Kevin T ; Maccoss, Malcolm ; Thornberry, Nancy A ; Peterson, Erin P

Bioorganic & Medicinal Chemistry Letters, 1994, Vol.4(16), pp.1965-1968 [Peer Reviewed Journal]

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18
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Administration of a HepDirect™ Prodrug of 2′-C-methylcytidine to Hepatitis C Virus Infected Chimpanzees

Carroll, Steven ; Koeplinger, Kenneth ; Vavrek, Marissa ; Handt, Laurence ; Maccoss, Malcolm ; Hecker, Scott ; Olsen, David

Antiviral Research, May 2009, Vol.82(2), pp.A22-A22 [Peer Reviewed Journal]

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19
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Alpha-aminothiazole-gamma-aminobutanoic amides as potent, small molecule CCR2 receptor antagonists

Zhou, Changyou ; Guo, Liangqin ; Parsons, William H ; Mills, Sander G ; Maccoss, Malcolm ; Vicario, Pasquale P ; Zweerink, Hans ; Cascieri, Margaret A ; Springer, Martin S ; Yang, Lihu

Bioorganic & medicinal chemistry letters, 15 January 2007, Vol.17(2), pp.309-14 [Peer Reviewed Journal]

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20
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Amidines as amide bond replacements in VLA-4 antagonists

Kamenecka, Theodore M ; Park, You-Jung ; Lin, Linus S ; de Laszlo, Stephen ; Mccauley, Ermengilda D ; Van Riper, Gail ; Egger, Linda ; Kidambi, Usha ; Mumford, Richard A ; Tong, Sharon ; Tang, Wei ; Colletti, Adria ; Teffera, Yohannes ; Stearns, Ralph ; Maccoss, Malcolm ; Schmidt, John A ; Hagmann, William K

Bioorganic & Medicinal Chemistry Letters, 03 May 2004, Vol.14(9), pp.2323-2326 [Peer Reviewed Journal]

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21
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An expeditious synthesis of 3-(difluoromethoxy)- and 3-(trifluoromethoxy)-5,6,7,8-tetrahydro-1,6-naphthyridines

Guiadeen, Deodialsingh ; Kothandaraman, Shankaran ; Yang, Lihu ; Mills, Sander G ; Maccoss, Malcolm

Tetrahedron Letters, 2008, Vol.49(44), pp.6368-6370 [Peer Reviewed Journal]

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22
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Antagonists of the human CCR5 receptor as anti-HIV-1 agents. Part 2: structure–activity relationships for substituted 2-aryl-1-[N-(methyl)-N-(phenylsulfonyl)amino]-4-(piperidin-1-yl)butanes

Finke, Paul E ; Meurer, Laura C ; Oates, Bryan ; Mills, Sander G ; Maccoss, Malcolm ; Malkowitz, Lorraine ; Springer, Martin S ; Daugherty, Bruce L ; Gould, Sandra L ; Demartino, Julie A ; Siciliano, Salvatore J ; Carella, Anthony ; Carver, Gwen ; Holmes, Karen ; Danzeisen, Renee ; Hazuda, Daria ; Kessler, Joseph ; Lineberger, Janet ; Miller, Michael ; Schleif, William A ; Emini, Emilio A

Bioorganic & Medicinal Chemistry Letters, January 2001, Vol.11(2), pp.265-270 [Peer Reviewed Journal]

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23
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Antagonists of the human CCR5 receptor as anti-HIV-1 agents. Part 4: synthesis and structure–Activity relationships for 1-[ N-(Methyl)- N-(phenylsulfonyl)amino]-2-(phenyl)-4-(4-( N-(alkyl)- N-(benzyloxycarbonyl)amino)piperidin-1-yl)butanes

Finke, Paul E ; Oates, Bryan ; Mills, Sander G ; Maccoss, Malcolm ; Malkowitz, Lorraine ; Springer, Martin S ; Gould, Sandra L ; Demartino, Julie A ; Carella, Anthony ; Carver, Gwen ; Holmes, Karen ; Danzeisen, Renee ; Hazuda, Daria ; Kessler, Joseph ; Lineberger, Janet ; Miller, Michael ; Schleif, William A ; Emini, Emilio A

Bioorganic & Medicinal Chemistry Letters, 2001, Vol.11(18), pp.2475-2479 [Peer Reviewed Journal]

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24
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Antiviral efficacy upon administration of a HepDirect prodrug of 2'-C-methylcytidine to hepatitis C virus-infected chimpanzees

Carroll, Steven S ; Koeplinger, Kenneth ; Vavrek, Marissa ; Zhang, Nanyan Rena ; Handt, Laurence ; Maccoss, Malcolm ; Olsen, David B ; Reddy, K Raja ; Sun, Zhili ; Van Poelje, Paul D ; Fujitaki, James M ; Boyer, Serge H ; Linemeyer, David L ; Hecker, Scott J ; Erion, Mark D

Antimicrobial agents and chemotherapy, August 2011, Vol.55(8), pp.3854-60 [Peer Reviewed Journal]

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25
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Bicyclic amidine inhibitors of nitric oxide synthase: discovery of perhydro-iminopyrindine and perhydro-iminoquinoline as potent, orally active inhibitors of inducible nitric oxide synthase

Guthikonda, Ravindra N ; Shah, Shrenik K ; Pacholok, Stephen G ; Humes, John L ; Mumford, Richard A ; Grant, Stephan K ; Chabin, Renee M ; Green, Barbara G ; Tsou, Nancy ; Ball, Richard ; Fletcher, Daniel S ; Luell, Silvi ; Euan Macintyre, D ; Maccoss, Malcolm

Bioorganic & Medicinal Chemistry Letters, 2005, Vol.15(8), pp.1997-2001 [Peer Reviewed Journal]

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26
Binding of 2-Aryl-4-(piperidin-1-yl)butanamines and 1,3,4-Trisubstituted Pyrrolidines to Human CCR5:  A Molecular Modeling-Guided Mutagenesis Study of the Binding Pocket
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Binding of 2-Aryl-4-(piperidin-1-yl)butanamines and 1,3,4-Trisubstituted Pyrrolidines to Human CCR5:  A Molecular Modeling-Guided Mutagenesis Study of the Binding Pocket

Castonguay, Laurie A. ; Weng, Youmin ; Adolfsen, William ; Di Salvo, Jerry ; Kilburn, Ruth ; Caldwell, Charles G. ; Daugherty, Bruce L. ; Finke, Paul E. ; Hale, Jeffrey J. ; Lynch, Christopher L. ; Mills, Sander G. ; Maccoss, Malcolm ; Springer, Martin S. ; Demartino, Julie A.

Biochemistry, 02/2003, Vol.42(6), pp.1544-1550 [Peer Reviewed Journal]

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27
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Bioisosteric replacement of anilide with benzoxazole: potent and orally bioavailable antagonists of VLA-4

Lin, Linus S ; Lanza, Thomas J ; Castonguay, Laurie A ; Kamenecka, Theodore ; Mccauley, Ermenegilda ; Van Riper, Gail ; Egger, Linda A ; Mumford, Richard A ; Tong, Xinchun ; Maccoss, Malcolm ; Schmidt, John A ; Hagmann, William K

Bioorganic & Medicinal Chemistry Letters, 03 May 2004, Vol.14(9), pp.2331-2334 [Peer Reviewed Journal]

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28
CCR5 Antagonists: 3-(Pyrrolidin-1-yl)propionic Acid Analogues with Potent Anti-HIV Activity
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CCR5 Antagonists: 3-(Pyrrolidin-1-yl)propionic Acid Analogues with Potent Anti-HIV Activity

Lynch, Christopher L. ; Hale, Jeffrey J. ; Budhu, Richard J. ; Gentry, Amy L. ; Finke, Paul E. ; Caldwell, Charles G. ; Mills, Sander G. ; Maccoss, Malcolm ; Shen, Dong-Ming ; Chapman, Kevin T. ; Malkowitz, Lorraine ; Springer, Martin S. ; Gould, Sandra L. ; Demartino, Julie A. ; Siciliano, Salvatore J. ; Cascieri, Margaret A. ; Carella, Anthony ; Carver, Gwen ; Holmes, Karen ; Schleif, William A. ; Danzeisen, Renee ; Hazuda, Daria ; Kessler, Joseph ; Lineberger, Janet ; Miller, Michael ; Emini, Emilio

Organic Letters, 07/2003, Vol.5(14), pp.2473-2475 [Peer Reviewed Journal]

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29
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CCR5 antagonists: bicyclic isoxazolidines as conformationally constrained N-1-substituted pyrrolidines

Lynch, Christopher L ; Gentry, Amy L ; Hale, Jeffrey J ; Mills, Sander G ; Maccoss, Malcolm ; Malkowitz, Lorraine ; Springer, Martin S ; Gould, Sandra L ; Demartino, Julie A ; Siciliano, Salvatore J ; Cascieri, Margaret A ; Doss, George ; Carella, Anthony ; Carver, Gwen ; Holmes, Karen ; Schleif, William A ; Danzeisen, Renee ; Hazuda, Daria ; Kessler, Joseph ; Lineberger, Janet ; Miller, Michael ; Emini, Emilio A

Bioorganic & Medicinal Chemistry Letters, 2002, Vol.12(4), pp.677-679 [Peer Reviewed Journal]

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30
C−H Cyanation of 6-Ring N-Containing Heteroaromatics
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C−H Cyanation of 6-Ring N-Containing Heteroaromatics

Elbert, Bryony L. ; Farley, Alistair J. M. ; Gorman, Timothy W. ; Johnson, Tarn C. ; Genicot, Christophe ; Lallemand, Bénédicte ; Pasau, Patrick ; Flasz, Jakub ; Castro, José L. ; Maccoss, Malcolm ; Paton, Robert S. ; Schofield, Christopher J. ; Smith, Martin D. ; Willis, Michael C. ; Dixon, Darren J.

Chemistry - A European Journal, 10/20/2017, Vol.23(59), pp.14733-14737 [Peer Reviewed Journal]

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31
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Characterization of resistance to non-obligate chain-terminating ribonucleoside analogs that inhibit hepatitis C virus replication in vitro

Migliaccio, Giovanni ; Tomassini, Joanne E ; Carroll, Steven S ; Tomei, Licia ; Altamura, Sergio ; Bhat, Balkrishen ; Bartholomew, Linda ; Bosserman, Michele R ; Ceccacci, Alessandra ; Colwell, Lawrence F ; Cortese, Riccardo ; De Francesco, Raffaele ; Eldrup, Anne B ; Getty, Krista L ; Hou, Xiaoli S ; Lafemina, Robert L ; Ludmerer, Steven W ; Maccoss, Malcolm ; Mcmasters, Daniel R ; Stahlhut, Mark W ; Olsen, David B ; Hazuda, Daria J ; Flores, Osvaldo A

The Journal of biological chemistry, 05 December 2003, Vol.278(49), pp.49164-70 [Peer Reviewed Journal]

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32
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Combining Molecular Scaffolds from FDA Approved Drugs: Application to Drug Discovery

Taylor, Richard D ; Maccoss, Malcolm ; Lawson, Alastair D G

Journal of medicinal chemistry, 09 March 2017, Vol.60(5), pp.1638-1647 [Peer Reviewed Journal]

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33
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Concise preparation of 8-trifluoromethyltetrahydro-6 H-pyrido [1,2- a] pyrazine-6-one

Kothandaraman, Shankaran ; Guiadeen, Deodialsingh ; Butora, Gabor ; Doss, George ; Mills, Sander G ; Maccoss, Malcolm ; Yang, Lihu

Tetrahedron Letters, 2009, Vol.50(28), pp.4050-4053 [Peer Reviewed Journal]

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34
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CorrigendumCorrigendum to “The discovery of acylated β-Amino acids as potent and orally bioavailable VLA-4 antagonists”[Bioorg. Med. Chem. Lett. 12 (2002) 611]

Lin, Linus S ; Kopka, Ihor E ; Mumford, Richard A ; Magriotis, Plato A ; Lanza, Jr, Thomas ; Durette, Philippe L ; Kamenecka, Theodore ; Young, David N ; de Laszlo, Stephen E ; Mccauley, Ermenegilda ; Van Riper, Gail ; Kidambi, Usha ; Egger, Linda A ; Tong, Xinchun ; Lyons, Kathryn ; Vincent, Stella ; Stearns, Ralph ; Colletti, Adria ; Teffera, Yohannes ; Fenyk-Melody, Judy ; Schmidt, John A ; Maccoss, Malcolm ; Hagmann, William K

Bioorganic & Medicinal Chemistry Letters, 2002, Vol.12(12), pp.1695-1695 [Peer Reviewed Journal]

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35
Cyclic Hydroxyamidines as Amide Isosteres: Discovery of Oxadiazolines and Oxadiazines as Potent and Highly Efficacious γ-Secretase Modulators in Vivo
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Cyclic Hydroxyamidines as Amide Isosteres: Discovery of Oxadiazolines and Oxadiazines as Potent and Highly Efficacious γ-Secretase Modulators in Vivo

Sun, Zhong-Yue ; Asberom, Theodros ; Bara, Thomas ; Bennett, Chad ; Burnett, Duane ; Chu, Inhou ; Clader, John ; Cohen-Williams, Mary ; Cole, David ; Czarniecki, Michael ; Durkin, James ; Gallo, Gioconda ; Greenlee, William ; Josien, Hubert ; Huang, Xianhai ; Hyde, Lynn ; Jones, Nicholas ; Kazakevich, Irina ; Li, Hongmei ; Liu, Xiaoxiang ; Lee, Julie ; Maccoss, Malcolm ; Mandal, Mihir B. ; Mccracken, Troy ; Nomeir, Amin ; Mazzola, Robert ; Palani, Anandan ; Parker, Eric M. ; Pissarnitski, Dmitri A. ; Qin, Jun ; Song, Lixin ; Terracina, Giuseppe ; Vicarel, Monica ; Voigt, Johannes ; Xu, Ruo ; Zhang, Lili ; Zhang, Qi ; Zhao, Zhiqiang ; Zhu, Xiaohong ; Zhu, Zhaoning

Journal of Medicinal Chemistry, 01/12/2012, Vol.55(1), pp.489-502 [Peer Reviewed Journal]

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