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Importance of Rigidity in Designing Small Molecule Drugs To Tackle Protein-Protein Interactions (PPIs) through Stabilization of Desired Conformers

Lawson, Alastair D G ; Maccoss, Malcolm ; Heer, Jag P

Journal of medicinal chemistry, 24 May 2018, Vol.61(10), pp.4283-4289 [Peer Reviewed Journal]

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Direct sulfonylation of anilines mediated by visible light † †Electronic supplementary information (ESI) available. See DOI: 10.1039/c7sc03891g

Johnson, Tarn C ; Elbert, Bryony l ; Farley, Alistair J. M ; Gorman, Timothy W ; Genicot, Christophe ; Lallemand, Bénédicte ; Pasau, Patrick ; Flasz, Jakub ; Castro, José L ; Maccoss, Malcolm ; Dixon, Darren J ; Paton, Robert S ; Schofield, Christopher J ; Smith, Martin D ; Willis, Michael C

Chemical Science, 2017, Vol.9(3), p.629-633 [Peer Reviewed Journal]

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C−H Cyanation of 6‐Ring N‐Containing Heteroaromatics

Elbert, Bryony L ; Farley, Alistair J. M ; Gorman, Timothy W ; Johnson, Tarn C ; Genicot, Christophe ; Lallemand, Bénédicte ; Pasau, Patrick ; Flasz, Jakub ; Castro, José L ; Maccoss, Malcolm ; Paton, Robert S ; Schofield, Christopher J ; Smith, Martin D ; Willis, Michael C ; Dixon, Darren J

Chemistry (Weinheim an Der Bergstrasse, Germany), 2017, Vol.23(59), p.14733-14737 [Peer Reviewed Journal]

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Combining Molecular Scaffolds from FDA Approved Drugs: Application to Drug Discovery

Taylor, Richard D ; Maccoss, Malcolm ; Lawson, Alastair D G

Journal of medicinal chemistry, 09 March 2017, Vol.60(5), pp.1638-1647 [Peer Reviewed Journal]

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Rings in drugs

Taylor, Richard D ; Maccoss, Malcolm ; Lawson, Alastair D G

Journal of medicinal chemistry, 24 July 2014, Vol.57(14), pp.5845-59 [Peer Reviewed Journal]

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Synthesis and SAR of geminal substitutions at the C5′ carbosugar position of pyrimidine-derived HCV inhibitors
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Synthesis and SAR of geminal substitutions at the C5′ carbosugar position of pyrimidine-derived HCV inhibitors

Verma, Vishal A. ; Rossman, Randall ; Bennett, Frank ; Chen, Lei ; Gavalas, Stephen ; Girijavallabhan, Vinay ; Huang, Yuhua ; Kim, Seong-Heon ; Kosinski, Aneta ; Pinto, Patrick ; Rizvi, Razia ; Shankar, Bandarpalle ; Tong, Ling ; Velazquez, Francisco ; Venkatraman, Srikanth ; Kozlowski, Joseph ; Maccoss, Malcolm ; Kwong, Cecil D. ; Bansal, Namita ; Kezar, Hollis S. ; Reynolds, Robert C. ; Maddry, Joseph A. ; Ananthan, Subramaniam ; Secrist, John A. ; Li, Cheng ; Chase, Robert ; Curry, Stephanie ; Huang, Hsueh-Cheng ; Tong, Xiao ; Njoroge, F. George ; Arasappan, Ashok

Bioorganic & Medicinal Chemistry Letters, 11/2012, Vol.22(22), pp.6967-6973 [Peer Reviewed Journal]

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Synthesis and SAR of pyridothiazole substituted pyrimidine derived HCV replication inhibitors
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Synthesis and SAR of pyridothiazole substituted pyrimidine derived HCV replication inhibitors

Girijavallabhan, Vinay M. ; Alvarez, Carmen ; Bennett, Frank ; Chen, Lei ; Gavalas, Stephen ; Huang, Yuhua ; Kim, Seong-Heon ; Kosinski, Aneta ; Pinto, Patrick ; Rizvi, Razia ; Rossman, Randall ; Shankar, Bandarpalle ; Tong, Ling ; Velazquez, Francisco ; Venkatraman, Srikanth ; Verma, Vishal A. ; Kozlowski, Joseph ; Shih, Neng-Yang ; Piwinski, John J. ; Maccoss, Malcolm ; Kwong, Cecil D. ; Bansal, Namita ; Clark, Jeremy L. ; Fowler, Anita T. ; Kezar, Hollis S. ; Valiyaveettil, Jacob ; Reynolds, Robert C. ; Maddry, Joseph A. ; Ananthan, Subramaniam ; Secrist, John A. ; Li, Cheng ; Chase, Robert ; Curry, Stephanie ; Huang, Hsueh-Cheng ; Tong, Xiao ; Njoroge, F. George ; Arasappan, Ashok

Bioorganic & Medicinal Chemistry Letters, 09/2012, Vol.22(17), pp.5652-5657 [Peer Reviewed Journal]

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Pyridofuran substituted pyrimidine derivatives as HCV replication (replicase) inhibitors
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Pyridofuran substituted pyrimidine derivatives as HCV replication (replicase) inhibitors

Bennett, Frank ; Kezar, Hollis S. ; Girijavallabhan, Vinay ; Huang, Yuhua ; Huelgas, Regina ; Rossman, Randall ; Shih, Neng-Yang ; Piwinski, John J. ; Maccoss, Malcolm ; Kwong, Cecil D. ; Clark, Jeremy L. ; Fowler, Anita T. ; Geng, Feng ; Roychowdhury, Abhijit ; Reynolds, Robert C. ; Maddry, Joseph A. ; Ananthan, Subramaniam ; Secrist, John A. ; Li, Cheng ; Chase, Robert ; Curry, Stephanie ; Huang, Hsueh-Cheng ; Tong, Xiao ; George Njoroge, F. ; Arasappan, Ashok

Bioorganic & Medicinal Chemistry Letters, 8/2012, Vol.22(15), pp.5144-5149 [Peer Reviewed Journal]

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A notable conversion of a thiolacetate to its corresponding sulfonyl chloride
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A notable conversion of a thiolacetate to its corresponding sulfonyl chloride

Huang, Yuhua ; Bennett, Frank ; Verma, Vishal ; George Njoroge, F. ; Maccoss, Malcolm

Tetrahedron Letters, 06/2012, Vol.53(26), pp.3203-3205 [Peer Reviewed Journal]

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5-Benzothiazole substituted pyrimidine derivatives as HCV replication (replicase) inhibitors
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5-Benzothiazole substituted pyrimidine derivatives as HCV replication (replicase) inhibitors

Arasappan, Ashok ; Bennett, Frank ; Girijavallabhan, Vinay ; Huang, Yuhua ; Huelgas, Regina ; Alvarez, Carmen ; Chen, Lei ; Gavalas, Stephen ; Kim, Seong-Heon ; Kosinski, Aneta ; Pinto, Patrick ; Rizvi, Razia ; Rossman, Randall ; Shankar, Bandarpalle ; Tong, Ling ; Velazquez, Francisco ; Venkatraman, Srikanth ; Verma, Vishal A. ; Kozlowski, Joseph ; Shih, Neng-Yang ; Piwinski, John J. ; Maccoss, Malcolm ; Kwong, Cecil D. ; Clark, Jeremy L. ; Fowler, Anita T. ; Geng, Feng ; Kezar, Hollis S. ; Roychowdhury, Abhijit ; Reynolds, Robert C. ; Maddry, Joseph A. ; Ananthan, Subramaniam ; Secrist, John A. ; Li, Cheng ; Chase, Robert ; Curry, Stephanie ; Huang, Hsueh-Cheng ; Tong, Xiao ; Njoroge, F. George

Bioorganic & Medicinal Chemistry Letters, 05/2012, Vol.22(9), pp.3229-3234 [Peer Reviewed Journal]

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Cyclic hydroxyamidines as amide isosteres: discovery of oxadiazolines and oxadiazines as potent and highly efficacious γ-secretase modulators in vivo

Sun, Zhong-Yue ; Asberom, Theodros ; Bara, Thomas ; Bennett, Chad ; Burnett, Duane ; Chu, Inhou ; Clader, John ; Cohen-Williams, Mary ; Cole, David ; Czarniecki, Michael ; Durkin, James ; Gallo, Gioconda ; Greenlee, William ; Josien, Hubert ; Huang, Xianhai ; Hyde, Lynn ; Jones, Nicholas ; Kazakevich, Irina ; Li, Hongmei ; Liu, Xiaoxiang ; Lee, Julie ; Maccoss, Malcolm ; Mandal, Mihir B ; Mccracken, Troy ; Nomeir, Amin ; Mazzola, Robert ; Palani, Anandan ; Parker, Eric M ; Pissarnitski, Dmitri A ; Qin, Jun ; Song, Lixin ; Terracina, Giuseppe ; Vicarel, Monica ; Voigt, Johannes ; Xu, Ruo ; Zhang, Lili ; Zhang, Qi ; Zhao, Zhiqiang ; Zhu, Xiaohong ; Zhu, Zhaoning

Journal of medicinal chemistry, 12 January 2012, Vol.55(1), pp.489-502 [Peer Reviewed Journal]

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Antiviral efficacy upon administration of a HepDirect prodrug of 2'-C-methylcytidine to hepatitis C virus-infected chimpanzees

Carroll, Steven S ; Koeplinger, Kenneth ; Vavrek, Marissa ; Zhang, Nanyan Rena ; Handt, Laurence ; Maccoss, Malcolm ; Olsen, David B ; Reddy, K Raja ; Sun, Zhili ; Van Poelje, Paul D ; Fujitaki, James M ; Boyer, Serge H ; Linemeyer, David L ; Hecker, Scott J ; Erion, Mark D

Antimicrobial agents and chemotherapy, August 2011, Vol.55(8), pp.3854-60 [Peer Reviewed Journal]

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Sustained viral response in a hepatitis C virus-infected chimpanzee via a combination of direct-acting antiviral agents

Olsen, David B ; Davies, Mary-Ellen ; Handt, Larry ; Koeplinger, Kenneth ; Zhang, Nanyan Rena ; Ludmerer, Steven W ; Graham, Donald ; Liverton, Nigel ; Maccoss, Malcolm ; Hazuda, Daria ; Carroll, Steven S

Antimicrobial agents and chemotherapy, February 2011, Vol.55(2), pp.937-9 [Peer Reviewed Journal]

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14
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Novel methods to functionalize thiazolo[4,5- c]pyridines

Girijavallabhan, Vinay ; Arasappan, Ashok ; Bennett, Frank ; Huang, Yuhua ; George Njoroge, F ; Maccoss, Malcolm

Tetrahedron Letters, 2010, Vol.51(21), pp.2797-2799 [Peer Reviewed Journal]

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15
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Syntheses of 4- and 6-substituted thiazolo[4,5- c]pyridines

Huang, Yuhua ; Bennett, Frank ; Girijavallabhan, Vinay ; Alvarez, Carmen ; Chan, Tze-Ming ; Osterman, Rebecca ; Senior, Mary ; Kwong, Cecil ; Bansal, Namita ; George Njoroge, F ; Maccoss, Malcolm

Tetrahedron Letters, 2010, Vol.51(21), pp.2800-2802 [Peer Reviewed Journal]

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16
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Phosphoramidate prodrugs of 2'-C-methylcytidine for therapy of hepatitis C virus infection

Gardelli, Cristina ; Attenni, Barbara ; Donghi, Monica ; Meppen, Malte ; Pacini, Barbara ; Harper, Steven ; Di Marco, Annalise ; Fiore, Fabrizio ; Giuliano, Claudio ; Pucci, Vincenzo ; Laufer, Ralph ; Gennari, Nadia ; Marcucci, Isabella ; Leone, Joseph F ; Olsen, David B ; Maccoss, Malcolm ; Rowley, Michael ; Narjes, Frank

Journal of medicinal chemistry, 10 September 2009, Vol.52(17), pp.5394-407 [Peer Reviewed Journal]

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Discovery of N-{N-(3-cyanophenyl)sulfonyl-4(R)-cyclobutylamino-(L)-prolyl}-4-(3',5'-dichloroisonicotinoyl) amino-(L)-phenylalanine (MK-0668), an extremely potent and orally active antagonist of very late antigen-4

Lin, Linus S ; Lanza, Thomas ; Jewell, James P ; Liu, Ping ; Jones, Carrie ; Kieczykowski, Gerard R ; Treonze, Kelly ; Si, Qian ; Manior, Salony ; Koo, Gloria ; Tong, Xinchun ; Wang, Junying ; Schuelke, Anne ; Pivnichny, James ; Wang, Regina ; Raab, Conrad ; Vincent, Stella ; Davies, Philip ; Maccoss, Malcolm ; Mumford, Richard A ; Hagmann, William K

Journal of medicinal chemistry, 11 June 2009, Vol.52(11), pp.3449-52 [Peer Reviewed Journal]

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18
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Administration of a HepDirect™ Prodrug of 2′-C-methylcytidine to Hepatitis C Virus Infected Chimpanzees

Carroll, Steven ; Koeplinger, Kenneth ; Vavrek, Marissa ; Handt, Laurence ; Maccoss, Malcolm ; Hecker, Scott ; Olsen, David

Antiviral Research, May 2009, Vol.82(2), pp.A22-A22 [Peer Reviewed Journal]

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19
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Robust antiviral efficacy upon administration of a nucleoside analog to hepatitis C virus-infected chimpanzees

Carroll, Steven S ; Ludmerer, Steven ; Handt, Larry ; Koeplinger, Kenneth ; Zhang, Nanyan Rena ; Graham, Donald ; Davies, Mary-Ellen ; Maccoss, Malcolm ; Hazuda, Daria ; Olsen, David B

Antimicrobial agents and chemotherapy, March 2009, Vol.53(3), pp.926-34 [Peer Reviewed Journal]

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20
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Concise preparation of 8-trifluoromethyltetrahydro-6 H-pyrido [1,2- a] pyrazine-6-one

Kothandaraman, Shankaran ; Guiadeen, Deodialsingh ; Butora, Gabor ; Doss, George ; Mills, Sander G ; Maccoss, Malcolm ; Yang, Lihu

Tetrahedron Letters, 2009, Vol.50(28), pp.4050-4053 [Peer Reviewed Journal]

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21
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Synthesis and biological evaluation of platensimycin analogs

Shen, Hong C ; Ding, Fa-Xiang ; Singh, Sheo B ; Parthasarathy, Gopalakrishnan ; Soisson, Stephen M ; Ha, Sookhee N ; Chen, Xun ; Kodali, Srinivas ; Wang, Jun ; Dorso, Karen ; Tata, James R ; Hammond, Milton L ; Maccoss, Malcolm ; Colletti, Steven L

Bioorganic & Medicinal Chemistry Letters, 2009, Vol.19(6), pp.1623-1627 [Peer Reviewed Journal]

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22
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Design, synthesis, and structure–activity relationship of novel CCR2 antagonists

Kothandaraman, Shankaran ; Donnely, Karla L ; Butora, Gabor ; Jiao, Richard ; Pasternak, Alexander ; Morriello, Gregori J ; Goble, Stephen D ; Zhou, Changyou ; Mills, Sander G ; Maccoss, Malcolm ; Vicario, Pasquale P ; Ayala, Julia M ; Demartino, Julie A ; Struthers, Mary ; Cascieri, Margaret A ; Yang, Lihu

Bioorganic & Medicinal Chemistry Letters, 2009, Vol.19(6), pp.1830-1834 [Peer Reviewed Journal]

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23
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An expeditious synthesis of 3-(difluoromethoxy)- and 3-(trifluoromethoxy)-5,6,7,8-tetrahydro-1,6-naphthyridines

Guiadeen, Deodialsingh ; Kothandaraman, Shankaran ; Yang, Lihu ; Mills, Sander G ; Maccoss, Malcolm

Tetrahedron Letters, 2008, Vol.49(44), pp.6368-6370 [Peer Reviewed Journal]

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24
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Synthesis of 2′-β- C-methyl-neplanocin derivatives as anti-HCV agents

Liao, Xibin ; Butora, Gabor ; Olsen, David B ; Carroll, Steven S ; Mcmasters, Daniel R ; Leone, Joseph F ; Stahlhut, Mark ; Doss, George A ; Yang, Lihu ; Maccoss, Malcolm

Tetrahedron Letters, 2008, Vol.49(26), pp.4149-4152 [Peer Reviewed Journal]

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25
Liver-Targeted Prodrugs of 2‘- C -Methyladenosine for Therapy of Hepatitis C Virus Infection
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Liver-Targeted Prodrugs of 2‘- C -Methyladenosine for Therapy of Hepatitis C Virus Infection

Hecker, Scott J. ; Reddy, K. Raja ; van Poelje, Paul D. ; Sun, Zhili ; Huang, Wenjian ; Varkhedkar, Vaibhav ; Reddy, M. Venkat ; Fujitaki, James M. ; Olsen, David B. ; Koeplinger, Kenneth A. ; Boyer, Serge H. ; Linemeyer, David L. ; Maccoss, Malcolm ; Erion, Mark D.

Journal of Medicinal Chemistry, 08/2007, Vol.50(16), pp.3891-3896 [Peer Reviewed Journal]

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26
Discovery of 3-Piperidinyl-1-cyclopentanecarboxamide as a Novel Scaffold for Highly Potent CC Chemokine Receptor 2 Antagonists
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Discovery of 3-Piperidinyl-1-cyclopentanecarboxamide as a Novel Scaffold for Highly Potent CC Chemokine Receptor 2 Antagonists

Yang, Lihu ; Butora, Gabor ; Jiao, Richard X. ; Pasternak, Alex ; Zhou, Changyou ; Parsons, William H. ; Mills, Sander G. ; Vicario, Pasquale P. ; Ayala, Julia M. ; Cascieri, Margaret A. ; Maccoss, Malcolm

Journal of Medicinal Chemistry, 05/2007, Vol.50(11), pp.2609-2611 [Peer Reviewed Journal]

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27
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Alpha-aminothiazole-gamma-aminobutanoic amides as potent, small molecule CCR2 receptor antagonists

Zhou, Changyou ; Guo, Liangqin ; Parsons, William H ; Mills, Sander G ; Maccoss, Malcolm ; Vicario, Pasquale P ; Zweerink, Hans ; Cascieri, Margaret A ; Springer, Martin S ; Yang, Lihu

Bioorganic & medicinal chemistry letters, 15 January 2007, Vol.17(2), pp.309-14 [Peer Reviewed Journal]

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28
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The elusive 8-fluoroadenosine: a simple non-enzymatic synthesis and characterization

Butora, Gabor ; Schmitt, Christoph ; Levorse, Dorothy A ; Streckfuss, Eric ; Doss, George A ; Maccoss, Malcolm

Tetrahedron, 2007, Vol.63(18), pp.3782-3789 [Peer Reviewed Journal]

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29
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Highly constrained bicyclic VLA-4 antagonists

Chang, Linda L ; Truong, Quang ; Doss, George A ; Maccoss, Malcolm ; Lyons, Kathryn ; Mccauley, Ermengilda ; Mumford, Richard ; Forrest, Gail ; Vincent, Stella ; Schmidt, John A ; Hagmann, William K

Bioorganic & Medicinal Chemistry Letters, 2007, Vol.17(3), pp.597-601 [Peer Reviewed Journal]

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30
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Synthesis and HCV inhibitory properties of 9-deaza- and 7,9-dideaza-7-oxa-2′- C-methyladenosine

Butora, Gabor ; Olsen, David B ; Carroll, Steven S ; Mcmasters, Daniel R ; Schmitt, Christoph ; Leone, Joseph F ; Stahlhut, Mark ; Burlein, Christine ; Maccoss, Malcolm

Bioorganic & Medicinal Chemistry, 2007, Vol.15(15), pp.5219-5229 [Peer Reviewed Journal]

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31
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α-Aminothiazole-γ-aminobutanoic amides as potent, small molecule CCR2 receptor antagonists

Zhou, Changyou ; Guo, Liangqin ; Parsons, William H ; Mills, Sander G ; Maccoss, Malcolm ; Vicario, Pasquale P ; Zweerink, Hans ; Cascieri, Margaret A ; Springer, Martin S ; Yang, Lihu

Bioorganic & Medicinal Chemistry Letters, 2007, Vol.17(2), pp.309-314 [Peer Reviewed Journal]

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32
4-Amino-2-alkyl-butyramides as small molecule CCR2 antagonists with favorable pharmacokinetic properties
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4-Amino-2-alkyl-butyramides as small molecule CCR2 antagonists with favorable pharmacokinetic properties

Butora, Gabor ; Morriello, Gregori J. ; Kothandaraman, Shankaran ; Guiadeen, Deodialsingh ; Pasternak, Alexander ; Parsons, William H. ; Maccoss, Malcolm ; Vicario, Pasquale P. ; Cascieri, Margaret A. ; Yang, Lihu

Bioorganic & Medicinal Chemistry Letters, 9/2006, Vol.16(18), pp.4715-4722 [Peer Reviewed Journal]

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33
Novel, Orally Bioavailable γ-Aminoamide CC Chemokine Receptor 2 (CCR2) Antagonists
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Novel, Orally Bioavailable γ-Aminoamide CC Chemokine Receptor 2 (CCR2) Antagonists

Pasternak, Alexander ; Marino, Dominick ; Vicario, Pasquale P. ; Ayala, Julia Marie ; Cascierri, Margaret A. ; Parsons, William ; Mills, Sander G. ; Maccoss, Malcolm ; Yang, Lihu

Journal of Medicinal Chemistry, 08/2006, Vol.49(16), pp.4801-4804 [Peer Reviewed Journal]

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34
Synthesis and Study of Alendronate Derivatives as Potential Prodrugs of Alendronate Sodium for the Treatment of Low Bone Density and Osteoporosis
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Synthesis and Study of Alendronate Derivatives as Potential Prodrugs of Alendronate Sodium for the Treatment of Low Bone Density and Osteoporosis

Vachal, Petr ; Hale, Jeffrey J. ; Lu, Zhe ; Streckfuss, Eric C. ; Mills, Sander G. ; Maccoss, Malcolm ; Yin, Daniel H. ; Algayer, Kimberly ; Manser, Kimberly ; Kesisoglou, Filippos ; Ghosh, Soumojeet ; Alani, Laman L.

Journal of Medicinal Chemistry, 06/2006, Vol.49(11), pp.3060-3063 [Peer Reviewed Journal]

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35
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Cyclopentane-based human NK1 antagonists. Part 1: Discovery and initial SAR

Finke, Paul E ; Meurer, Laura C ; Levorse, Dorothy A ; Mills, Sander G ; Maccoss, Malcolm ; Sadowski, Sharon ; Cascieri, Margaret A ; Tsao, Kwei-Lan ; Chicchi, Gary G ; Metzger, Joseph M ; Macintyre, D. Euan

Bioorganic & Medicinal Chemistry Letters, 2006, Vol.16(17), pp.4497-4503 [Peer Reviewed Journal]

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