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Material Type: Article
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Identification of potent and selective amidobipyridyl inhibitors of protein kinase DMeredith, Erik L ; Beattie, Kimberly ; Burgis, Robin ; Capparelli, Michael ; Chapo, Joseph ; Dipietro, Lucian ; Gamber, Gabriel ; Enyedy, Istvan ; Hood, David B ; Hosagrahara, Vinayak ; Jewell, Charles ; Koch, Keith A ; Lee, Wendy ; Lemon, Douglas D ; Mckinsey, Timothy A ; Miranda, Karl ; Pagratis, Nikos ; Phan, Dillon ; Plato, Craig ; Rao, Chang ; Rozhitskaya, Olga ; Soldermann, Nicolas ; Springer, Clayton ; Van Eis, Maurice ; Vega, Richard B ; Yan, Wanlin ; Zhu, Qingming ; Monovich, Lauren GJournal of medicinal chemistry, 12 August 2010, Vol.53(15), pp.5422-38 [Peer Reviewed Journal]Full text available |
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Material Type: Article
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Identification of orally available naphthyridine protein kinase D inhibitorsMeredith, Erik L ; Ardayfio, Ophelia ; Beattie, Kimberly ; Dobler, Markus R ; Enyedy, Istvan ; Gaul, Christoph ; Hosagrahara, Vinayak ; Jewell, Charles ; Koch, Keith ; Lee, Wendy ; Lehmann, Hansjoerg ; Mckinsey, Timothy A ; Miranda, Karl ; Pagratis, Nikos ; Pancost, Margaret ; Patnaik, Anup ; Phan, Dillon ; Plato, Craig ; Qian, Ming ; Rajaraman, Vasumathy ; Rao, Chang ; Rozhitskaya, Olga ; Ruppen, Thomas ; Shi, Jie ; Siska, Sarah J ; Springer, Clayton ; Van Eis, Maurice ; Vega, Richard B ; Von Matt, Anette ; Yang, Lihua ; Yoon, Taeyoung ; Zhang, Ji-Hu ; Zhu, Na ; Monovich, Lauren GJournal of medicinal chemistry, 12 August 2010, Vol.53(15), pp.5400-21 [Peer Reviewed Journal]Full text available |
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Material Type: Article
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( R )-3,3,3-Trifluoro-2-hydroxy-2-methylpropionamides Are Orally Active Inhibitors of Pyruvate Dehydrogenase KinaseAicher, Thomas D. ; Anderson, Robert C. ; Bebernitz, Gregory R. ; Coppola, Gary M. ; Jewell, Charles F. ; Knorr, Douglas C. ; Liu, Charles ; Sperbeck, Donald M. ; Brand, Leonard J. ; Strohschein, Robert J. ; Gao, Jiaping ; Vinluan, Christine C. ; Shetty, Suraj S. ; Dragland, Carol ; Kaplan, Emma L. ; Delgrande, Dominick ; Islam, Amin ; Liu, Xilin ; Lozito, Robert J. ; Maniara, Wieslawa M. ; Walter, R. Erik ; Mann, William R.Journal of Medicinal Chemistry, 07/1999, Vol.42(15), pp.2741-2746 [Peer Reviewed Journal]Full text available |